| # | Aladdin ID | Assay Type | Description | Organism | Compounds | Reference | BAO Format | Source | |
|---|---|---|---|---|---|---|---|---|---|
| 1. | ALA2409983 | A | Ratio of AUC in mouse blood in presence of P-gp inhibitor GF120918 to AUC in mouse blood at 5 mg/kg, po | Mus musculus | 1 | organism-based format | Scientific Literature | ||
| 2. | ALA2409986 | F | Antidiabetic activity in ob/ob mouse assessed as reduction in blood glucose level at 100 mg/kg, po bid for 5 days in presence of P-gp inhibitor GF120918 relative to control | Mus musculus | 2 | organism-based format | Scientific Literature | ||
| 3. | ALA2409987 | B | Activation of human recombinant AMPK alpha2beta2gamma3 | Homo sapiens | 2 | protein complex format | Scientific Literature | ||
| 4. | ALA2409988 | B | Activation of human recombinant AMPK alpha2beta2gamma1 | Homo sapiens | 4 | protein complex format | Scientific Literature | ||
| 5. | ALA2409989 | B | Activation of human recombinant AMPK alpha1beta2gamma1 | Homo sapiens | 2 | protein complex format | Scientific Literature | ||
| 6. | ALA2409990 | B | Activation of human recombinant AMPK alpha2beta1gamma1 | Homo sapiens | 1 | protein complex format | Scientific Literature | ||
| 7. | ALA2409991 | B | Activation of human recombinant AMPK alpha1beta1gamma3 | Homo sapiens | 1 | protein complex format | Scientific Literature | ||
| 8. | ALA2409992 | B | Activation of human recombinant AMPK alpha1beta1gamma2 | Homo sapiens | 1 | protein complex format | Scientific Literature | ||
| 9. | ALA2409995 | A | Oral bioavailability in mouse at 5 mg/kg | Mus musculus | 8 | organism-based format | Scientific Literature | ||
| 10. | ALA2409996 | A | Clearance in mouse at 1 mg/kg, iv | Mus musculus | 9 | organism-based format | Scientific Literature | ||
| 11. | ALA2409998 | A | AUC in mouse at 5 mg/kg, po | Mus musculus | 8 | organism-based format | Scientific Literature | ||
| 12. | ALA2409999 | A | Plasma protein binding in mouse | Mus musculus | 8 | cell-free format | Scientific Literature | ||
| 13. | ALA2410000 | P | Solubility of the compound | 9 | small-molecule physicochemical format | Scientific Literature | |||
| 14. | ALA2410001 | A | Permeability of the compound by PAMPA | 9 | assay format | Scientific Literature | |||
| 15. | ALA2410002 | B | Activation of human recombinant AMPK alpha1beta1gamma1 by FRET assay | Homo sapiens | 12 | protein complex format | Scientific Literature |
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