# | Aladdin ID | Assay Type | Description | Organism | Compounds | Reference | BAO Format | Source | |
---|---|---|---|---|---|---|---|---|---|
1. | ALA2412024 | Binding | Inhibition of human plasma kallikrein using benzyloxycarbonyl-Phe-Arg-7-amino-4-methylcoumarin as substrate at 50 uM by fluorescence microplate reader analysis | Homo sapiens | 12 | ALA2406965 | single protein format | Scientific Literature | |
2. | ALA2412026 | Binding | Competitive inhibition of human neutrophil elastase using N-methylsuccinyl-Ala-Ala-Pro-Val-7-amino-4-methylcoumarin as substrate by Lineweaver-Burk plot analysis | Homo sapiens | 2 | ALA2406965 | single protein format | Scientific Literature | |
3. | ALA2412027 | Binding | Inhibition of human neutrophil elastase using N-methylsuccinyl-Ala-Ala-Pro-Val-7-amino-4-methylcoumarin as substrate at 5 uM after 7 hrs by fluorescence microplate reader analysis | Homo sapiens | 1 | ALA2406965 | single protein format | Scientific Literature | |
4. | ALA2412029 | Binding | Inhibition of human neutrophil elastase using N-methylsuccinyl-Ala-Ala-Pro-Val-7-amino-4-methylcoumarin as substrate at 5 uM after 4 hrs by fluorescence microplate reader analysis | Homo sapiens | 5 | ALA2406965 | single protein format | Scientific Literature | |
5. | ALA2412030 | Physicochemical | Half life in phosphate buffer at pH 7.3 | 10 | ALA2406965 | small-molecule physicochemical format | Scientific Literature | ||
6. | ALA2412032 | Binding | Inhibition of human spleen cathepsin D using MOCAc-Gly-Lys-Pro-Ile-Leu-Phe-Phe-Arg-Leu-Lys (Dnp)-D-Arg-NH2 as substrate at 50 uM by fluorescence microplate reader analysis | Homo sapiens | 10 | ALA2406965 | single protein format | Scientific Literature | |
7. | ALA2412033 | Binding | Inhibition of human urokinase using benzyloxycarbonyl-Gly-Gly-Arg-7-amino-4-methylcoumarin as substrate by fluorescence microplate reader analysis | Homo sapiens | 9 | ALA2406965 | single protein format | Scientific Literature | |
8. | ALA2412035 | Binding | Inhibition of human neutrophil elastase using N-methylsuccinyl-Ala-Ala-Pro-Val-7-amino-4-methylcoumarin as substrate measured every 30 seconds for 10 mins by fluorescence microplate reader analysis | Homo sapiens | 42 | ALA2406965 | single protein format | Scientific Literature | |
9. | ALA2412036 | Binding | Inhibition of human pancreatic chymotrypsin using Suc-Ala-Ala-Pro-7-amino-4-methylcoumarin as substrate by fluorescence microplate reader analysis | Homo sapiens | 10 | ALA2406965 | single protein format | Scientific Literature | |
10. | ALA2412037 | Binding | Inhibition of human plasma thrombin using benzonyl-Phe-Val-Arg-7-amino-4-methylcoumarin as substrate by fluorescence microplate reader analysis | Homo sapiens | 10 | ALA2406965 | single protein format | Scientific Literature | |
11. | ALA4265084 | Binding | Inhibition of human neutrophil elastase using N-methylsuccinyl-Ala-Ala-Pro-Val-7-amino-4-methylcoumarin as substrate measured every 30 secs for 10 mins by fluorescence assay | Homo sapiens | 34 | ALA4261628 | single protein format | Scientific Literature |