| # | Aladdin ID | Assay Type | Description | Organism | Compounds | Reference | BAO Format | Source | |
|---|---|---|---|---|---|---|---|---|---|
| 1. | ALA2439932 | ADME | Fraction unbound in human | Homo sapiens | 2 | ALA2434833 | organism-based format | Scientific Literature | |
| 2. | ALA2439933 | ADME | Fraction unbound in mouse | Mus musculus | 2 | ALA2434833 | organism-based format | Scientific Literature | |
| 3. | ALA2439934 | ADME | Tmax in C57 mouse at 10 mg/kg, po | Mus musculus | 2 | ALA2434833 | organism-based format | Scientific Literature | |
| 4. | ALA2439935 | ADME | Oral bioavailability in C57 mouse at 10 mg/kg | Mus musculus | 2 | ALA2434833 | organism-based format | Scientific Literature | |
| 5. | ALA2439936 | Binding | Inhibition of human ERG | Homo sapiens | 2 | ALA2434833 | single protein format | Scientific Literature | |
| 6. | ALA2439937 | ADME | AUC in C57 mouse at 10 mg/kg, po | Mus musculus | 2 | ALA2434833 | organism-based format | Scientific Literature | |
| 7. | ALA2439938 | ADME | Cmax in C57 mouse at 10 mg/kg, po | Mus musculus | 2 | ALA2434833 | organism-based format | Scientific Literature | |
| 8. | ALA2439939 | ADME | Metabolic stability in human liver microsomes assessed as GSH adduct formation up to 10 uM relative to control | Homo sapiens | 2 | ALA2434833 | microsome format | Scientific Literature | |
| 9. | ALA2439941 | ADME | Inhibition of CYP2C9 (unknown origin) | Homo sapiens | 2 | ALA2434833 | single protein format | Scientific Literature | |
| 10. | ALA2439942 | ADME | Inhibition of CYP2D6 (unknown origin) | Homo sapiens | 2 | ALA2434833 | single protein format | Scientific Literature | |
| 11. | ALA2437633 | ADME | Ratio of Kinact to Ki for CYP3A4 in human liver microsomes | Homo sapiens | 10 | ALA2434833 | microsome format | Scientific Literature | |
| 12. | ALA2437634 | ADME | Time-dependent inhibition of CYP3A4 in human liver microsomes assessed as midazolam hydroxylation by LC-MS/MS analysis | Homo sapiens | 10 | ALA2434833 | microsome format | Scientific Literature | |
| 13. | ALA2437635 | ADME | Inhibition of CYP3A4 (unknown origin) | Homo sapiens | 35 | ALA2434833 | single protein format | Scientific Literature | |
| 14. | ALA2437636 | Binding | Displacement of AVPIAQKSEK (epsilon-biotin)-OH from 6xhistidine-thrombin-TEV-tagged XIAP BIR3 domain (241 to 356) (unknown origin) after 45 mins by TR-FRET Assay | Homo sapiens | 39 | ALA2434833 | single protein format | Scientific Literature | |
| 15. | ALA2437637 | Binding | Displacement of AVPIAQKSEK (epsilon-biotin)-OH from 6xhistidine-thrombin-TEV-tagged XIAP BIR2 domain (124 to 240) (unknown origin) after 45 mins by TR-FRET Assay | Homo sapiens | 39 | ALA2434833 | single protein format | Scientific Literature |
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