| # | Aladdin ID | Assay Type | Description | Organism | Compounds | Reference | BAO Format | Source | |
|---|---|---|---|---|---|---|---|---|---|
| 1. | ALA622143 | P | Calculated partition coefficient (clogP) | 22 | ALA1148355 | small-molecule physicochemical format | Scientific Literature | ||
| 2. | ALA685238 | B | Inhibitory activity against human Group IVA Phospholipase A2 (GIVA PLA2) | 3 | ALA1135491 | single protein format | Scientific Literature | ||
| 3. | ALA686432 | B | Mole fraction of compound in the total substrate interface required to inhibit human GIVA PLA2 by 50% | 10 | ALA1148355 | single protein format | Scientific Literature | ||
| 4. | ALA737120 | F | Tested on P388D1 macrophage-like cell line (AA-derived products) for inhibition of the GIVA PLA2 in the long-term lipopolysaccharide | Mus musculus | 1 | ALA1148355 | organism-based format | Scientific Literature | |
| 5. | ALA737121 | F | Tested on P388D1 macrophage-like cell line (PGE2 production) for inhibition of the GIVA PLA2 in the long-term lipopolysaccharide | Mus musculus | 1 | ALA1148355 | organism-based format | Scientific Literature | |
| 6. | ALA774974 | F | Compound was tested for in vivo analgesic activity in rat | Rattus norvegicus | 3 | ALA1148355 | organism-based format | Scientific Literature | |
| 7. | ALA782321 | F | Compound was tested for in vivo antiinflammatory activity in rat | Rattus norvegicus | 3 | ALA1148355 | organism-based format | Scientific Literature | |
| 8. | ALA861688 | B | Inhibition of group 6A iPLA2 at 0.091 mole fraction | Homo sapiens | 9 | ALA1147679 | single protein format | Scientific Literature | |
| 9. | ALA861689 | B | Inhibition of group 4A cPLA2 | Homo sapiens | 5 | ALA1147679 | single protein format | Scientific Literature | |
| 10. | ALA917108 | B | Inhibition of human cPLA2 alpha by GLU micelle assay | Homo sapiens | 37 | ALA1142935 | single protein format | Scientific Literature | |
| 11. | ALA917112 | F | Inhibition of A-23187-stimulated TXB2 production in Sprague-Dawley rat whole blood at 10 uM | Rattus norvegicus | 7 | ALA1142935 | tissue-based format | Scientific Literature | |
| 12. | ALA894459 | B | Inhibition of human GIVA cPLA2 | Homo sapiens | 21 | ALA1148742 | assay format | Scientific Literature | |
| 13. | ALA1042148 | F | Antiinflammatory activity in mouse RAW264.7 cells assessed as inhibition of Kdo2 lipid-A-stimulated arachidonic acid release after 1 hr | Mus musculus | 7 | ALA1154042 | cell-based format | Scientific Literature | |
| 14. | ALA1042149 | F | Antiinflammatory activity in mouse RAW264.7 cells assessed as inhibition of Kdo2 lipid-A-stimulated arachidonic acid release at 25 uM for 1 hr | Mus musculus | 21 | ALA1154042 | cell-based format | Scientific Literature | |
| 15. | ALA1948779 | B | Inhibition of cPLA2alpha | 19 | ALA1944552 | assay format | Scientific Literature | ||
| 16. | ALA4432418 | B | Inhibition of human group 6A iPLA2 using PAPC/[14C]-labeled PAPC as substrate at 0.091 mole fraction after 30 mins by mixed micelle-based assay relative to control | Homo sapiens | 10 | ALA4431346 | single protein format | Scientific Literature | |
| 17. | ALA4432422 | B | Inhibition of human group 4A cPLA2 using PAPC as substrate preincubated for 5 mins with substrate followed by enzyme addition for 30 mins by mixed micelle-based assay | Homo sapiens | 2 | ALA4431346 | single protein format | Scientific Literature |
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