| # | Aladdin ID | Assay Type | Description | Organism | Compounds | Reference | BAO Format | Source | |
|---|---|---|---|---|---|---|---|---|---|
| 1. | ALA3096226 | ADME | Metabolic stability in dog liver microsomes assessed as compound remaining at 4 uM after 30 mins by LC-ESI/MS analysis | Canis lupus familiaris | 26 | ALA3091283 | assay format | Scientific Literature | |
| 2. | ALA3096227 | ADME | Metabolic stability in rat liver microsomes assessed as compound remaining at 4 uM after 30 mins by LC-ESI/MS analysis | Rattus norvegicus | 26 | ALA3091283 | assay format | Scientific Literature | |
| 3. | ALA3096228 | ADME | Metabolic stability in human liver microsomes assessed as compound remaining at 4 uM after 30 mins by LC-ESI/MS analysis | Homo sapiens | 26 | ALA3091283 | assay format | Scientific Literature | |
| 4. | ALA3096229 | Binding | Displacement of [3H]-CP-55940 from rat CB2 receptor expressed in CHO cells after 90 mins | Rattus norvegicus | 26 | ALA3091283 | cell-based format | Scientific Literature | |
| 5. | ALA3096230 | Binding | Displacement of [3H]-CP-55940 from human CB2 receptor expressed in CHO cells after 90 mins | Homo sapiens | 26 | ALA3091283 | cell-based format | Scientific Literature | |
| 6. | ALA3096232 | Binding | Selectivity ratio of EC50 for human CB1 receptor to EC50 for human CB2 receptor | Homo sapiens | 25 | ALA3091283 | assay format | Scientific Literature | |
| 7. | ALA3096234 | Functional | Agonist activity at human CB1 receptor expressed in Sf9 cells assessed as stimulation of [35S]GTPgamma binding incubated for 15 mins prior to [35S]GTPgamma addition measured after 35 mins by scintillation proximity assay | Homo sapiens | 25 | ALA3091283 | cell-based format | Scientific Literature | |
| 8. | ALA3096235 | Functional | Agonist activity at human CB2 receptor expressed in CHO cells assessed as stimulation of [35S]GTPgamma binding after 30 mins by scintillation proximity assay relative to methanandamide | Homo sapiens | 26 | ALA3091283 | cell-based format | Scientific Literature | |
| 9. | ALA3096236 | Functional | Agonist activity at human CB2 receptor expressed in CHO cells assessed as stimulation of [35S]GTPgamma binding after 30 mins by scintillation proximity assay | Homo sapiens | 26 | ALA3091283 | cell-based format | Scientific Literature |
The page will load shortly, Thanks for your patience!