| # | Aladdin ID | Assay Type | Description | Organism | Compounds | Reference | BAO Format | Source | |
|---|---|---|---|---|---|---|---|---|---|
| 1. | ALA3105977 | B | Inhibition of rat recombinant 6xHis-tagged DYRK1A catalytic domain (1 to 502) expressed in Escherichia coli BL21 (DE3) using N-terminal fluorescein coupled KISGRLSPIMTEQ as substrate after 30 mins by HPLC analysis in presence of 50 uM ATP | Rattus norvegicus | 25 | assay format | Scientific Literature | ||
| 2. | ALA3371267 | F | Cell cycle arrest in human HMC-1.2 cells assessed as accumulation at G1 phase after 24 hrs by flow cytometric analysis | Homo sapiens | 1 | cell-based format | Scientific Literature | ||
| 3. | ALA3371268 | F | Induction of apoptosis in human HMC-1.2 cells assessed as apoptotic cells at 0.1 uM after 48 hrs by TUNEL staining (Rvb = 0.849%) | Homo sapiens | 1 | cell-based format | Scientific Literature | ||
| 4. | ALA3371269 | F | Induction of apoptosis in human HMC-1.2 cells assessed as apoptotic cells at 1 uM after 48 hrs by TUNEL staining (Rvb = 0.849%) | Homo sapiens | 1 | cell-based format | Scientific Literature | ||
| 5. | ALA3371270 | F | Induction of apoptosis in human HMC-1.2 cells assessed as apoptotic cells at 5 uM after 48 hrs by TUNEL staining (Rvb = 0.849%) | Homo sapiens | 1 | cell-based format | Scientific Literature | ||
| 6. | ALA3368317 | B | Inhibition of c-KIT D816V mutant (unknown origin) | Homo sapiens | 41 | single protein format | Scientific Literature | ||
| 7. | ALA3368318 | B | Inhibition of PI3Kalpha (unknown origin) | Homo sapiens | 20 | single protein format | Scientific Literature | ||
| 8. | ALA3368319 | B | Inhibition of wild type c-KIT (unknown origin) | Homo sapiens | 18 | single protein format | Scientific Literature | ||
| 9. | ALA3368320 | B | Inhibition of ABL T315I mutant (unknown origin) at 1 uM by KINOMEscanning assay relative to control | Homo sapiens | 5 | single protein format | Scientific Literature | ||
| 10. | ALA3368321 | B | Inhibition of AKT1 (unknown origin) at 1 uM by KINOMEscanning assay relative to control | Homo sapiens | 5 | single protein format | Scientific Literature | ||
| 11. | ALA3368322 | B | Inhibition of AKT2 (unknown origin) at 1 uM by KINOMEscanning assay relative to control | Homo sapiens | 5 | single protein format | Scientific Literature | ||
| 12. | ALA3368323 | B | Inhibition of ALK (unknown origin) at 1 uM by KINOMEscanning assay relative to control | Homo sapiens | 5 | single protein format | Scientific Literature | ||
| 13. | ALA3368324 | B | Inhibition of AMPKalpha 1 (unknown origin) at 1 uM by KINOMEscanning assay relative to control | Homo sapiens | 5 | single protein format | Scientific Literature | ||
| 14. | ALA3368325 | B | Inhibition of AMPKalpha 2 (unknown origin) at 1 uM by KINOMEscanning assay relative to control | Homo sapiens | 5 | single protein format | Scientific Literature | ||
| 15. | ALA3368326 | B | Inhibition of AURKA (unknown origin) at 1 uM by KINOMEscanning assay relative to control | Homo sapiens | 5 | single protein format | Scientific Literature | ||
| 16. | ALA3368327 | B | Inhibition of AURKB (unknown origin) at 1 uM by KINOMEscanning assay relative to control | Homo sapiens | 5 | single protein format | Scientific Literature | ||
| 17. | ALA3368328 | B | Inhibition of BRAF (unknown origin) at 1 uM by KINOMEscanning assay relative to control | Homo sapiens | 5 | single protein format | Scientific Literature | ||
| 18. | ALA3368329 | B | Inhibition of BRAF V600E mutant (unknown origin) at 1 uM by KINOMEscanning assay relative to control | Homo sapiens | 5 | single protein format | Scientific Literature | ||
| 19. | ALA3368330 | B | Inhibition of CAMK1 (unknown origin) at 1 uM by KINOMEscanning assay relative to control | Homo sapiens | 5 | single protein format | Scientific Literature | ||
| 20. | ALA3368331 | B | Inhibition of CDK4 (unknown origin) at 1 uM by KINOMEscanning assay relative to control | Homo sapiens | 5 | single protein format | Scientific Literature |
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