| # | Aladdin ID | Assay Type | Description | Organism | Compounds | Reference | BAO Format | Source | |
|---|---|---|---|---|---|---|---|---|---|
| 1. | ALA3123259 | F | Inverse agonist activity at human histamine H3 receptor by [35S]GTPgammaS binding assay | Homo sapiens | 2 | assay format | Scientific Literature | ||
| 2. | ALA3123306 | A | Ratio of drug uptake in brain to plasma in rat at 10 mg/kg, ip after 6 hrs | Rattus norvegicus | 2 | organism-based format | Scientific Literature | ||
| 3. | ALA3123309 | A | Oral bioavailability in rat at 5 mg/kg | Rattus norvegicus | 2 | organism-based format | Scientific Literature | ||
| 4. | ALA3123313 | A | Cmax in rat at 5 mg/kg, po | Rattus norvegicus | 2 | organism-based format | Scientific Literature | ||
| 5. | ALA3123316 | A | AUC in rat at 5 mg/kg, po | Rattus norvegicus | 2 | organism-based format | Scientific Literature | ||
| 6. | ALA3123319 | A | Clearance in rat at 1 mg/kg, iv | Rattus norvegicus | 2 | organism-based format | Scientific Literature | ||
| 7. | ALA3123321 | A | Volume of distribution at steady state in rat at 1 mg/kg, iv | Rattus norvegicus | 2 | organism-based format | Scientific Literature | ||
| 8. | ALA3123325 | A | Terminal half life in rat at 1 mg/kg, iv | Rattus norvegicus | 2 | organism-based format | Scientific Literature | ||
| 9. | ALA3123331 | B | Inhibition of human ERG channel by patch clamp technique | Homo sapiens | 2 | assay format | Scientific Literature | ||
| 10. | ALA3123333 | B | Inhibition of dopamine transporter (unknown origin) at 10 uM | Homo sapiens | 1 | single protein format | Scientific Literature | ||
| 11. | ALA3123334 | B | Inhibition of human histamine H4 receptor at 10 uM | Homo sapiens | 2 | single protein format | Scientific Literature | ||
| 12. | ALA3123335 | B | Inhibition of human histamine H1 receptor at 10 uM | Homo sapiens | 2 | single protein format | Scientific Literature | ||
| 13. | ALA3123336 | B | Inhibition of human histamine H2 receptor at 10 uM | Homo sapiens | 2 | single protein format | Scientific Literature | ||
| 14. | ALA3123337 | A | Half life in human liver microsomes | Homo sapiens | 2 | assay format | Scientific Literature | ||
| 15. | ALA3123338 | A | Half life in monkey liver microsomes | Macaca mulatta | 2 | microsome format | Scientific Literature | ||
| 16. | ALA3123339 | A | Half life in rat liver microsomes | Rattus norvegicus | 2 | assay format | Scientific Literature | ||
| 17. | ALA3123340 | A | Half life in dog liver microsomes | Canis lupus familiaris | 2 | assay format | Scientific Literature | ||
| 18. | ALA3123341 | A | Half life in mouse liver microsomes | Mus musculus | 2 | microsome format | Scientific Literature | ||
| 19. | ALA3123342 | A | Inhibition of CYP3A4 (unknown origin) | Homo sapiens | 4 | single protein format | Scientific Literature | ||
| 20. | ALA3123343 | A | Inhibition of CYP2D6 (unknown origin) | Homo sapiens | 4 | single protein format | Scientific Literature |
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