| # | Aladdin ID | Assay Type | Description | Organism | Compounds | Reference | BAO Format | Source | |
|---|---|---|---|---|---|---|---|---|---|
| 1. | ALA3132004 | F | In vivo inhibition of FAAH in C57Bl/6J mouse assessed as increase in OEA level in brain at 30 mg/kg, ip measured after > 6 hrs | Mus musculus | 2 | organism-based format | Scientific Literature | ||
| 2. | ALA3132005 | F | In vivo inhibition of FAAH in C57Bl/6J mouse assessed as increase in AEA level in brain at 30 mg/kg, ip measured after > 6 hrs | Mus musculus | 2 | organism-based format | Scientific Literature | ||
| 3. | ALA3132006 | F | In vivo inhibition of FAAH in C57Bl/6J mouse assessed as increase in PEA level in brain at 30 mg/kg, ip measured after > 6 hrs | Mus musculus | 2 | organism-based format | Scientific Literature | ||
| 4. | ALA3132007 | F | In vivo inhibition of FAAH in C57Bl/6J mouse assessed as increase in PEA level in brain at 30 mg/kg, ip measured within 1.5 to 3 hrs | Mus musculus | 2 | organism-based format | Scientific Literature | ||
| 5. | ALA3132008 | F | In vivo inhibition of FAAH in C57Bl/6J mouse assessed as increase in OEA level in brain at 30 mg/kg, ip measured within 1.5 to 3 hrs | Mus musculus | 2 | organism-based format | Scientific Literature | ||
| 6. | ALA3132009 | F | In vivo inhibition of FAAH in C57Bl/6J mouse assessed as increase in AEA level in brain at 30 mg/kg, ip measured within 1.5 to 3 hrs | Mus musculus | 2 | organism-based format | Scientific Literature | ||
| 7. | ALA3132010 | F | In vivo inhibition of FAAH in C57Bl/6J mouse assessed as increase in PEA level in brain at 30 mg/kg, ip after 3 hrs relative to vehicle-treated control | Mus musculus | 7 | organism-based format | Scientific Literature | ||
| 8. | ALA3132011 | F | In vivo inhibition of FAAH in C57Bl/6J mouse assessed as increase in OEA level in brain at 30 mg/kg, ip after 3 hrs relative to vehicle-treated control | Mus musculus | 7 | organism-based format | Scientific Literature | ||
| 9. | ALA3132012 | F | In vivo inhibition of FAAH in C57Bl/6J mouse assessed as increase in AEA level in brain at 30 mg/kg, ip after 3 hrs relative to vehicle-treated control | Mus musculus | 7 | organism-based format | Scientific Literature | ||
| 10. | ALA3132015 | B | Selectivity ratio of IC50 for mouse brain membrane MAGL to IC50 for mouse FAAH | Mus musculus | 6 | assay format | Scientific Literature | ||
| 11. | ALA3132016 | B | Selectivity ratio of IC50 for mouse brain membrane ABHD6 to IC50 for mouse FAAH | Mus musculus | 6 | assay format | Scientific Literature | ||
| 12. | ALA3132017 | B | Selectivity ratio of IC50 for mouse brain membrane KIAA1363 to IC50 for mouse FAAH | Mus musculus | 6 | assay format | Scientific Literature | ||
| 13. | ALA3129771 | B | Irreversible inhibition of recombinant rat FAAH expressed in Escherichia coli assessed as remaining activity at IC80 preincubated for 3 hrs followed by 370 fold dilution measured after 18 hrs | Rattus norvegicus | 8 | assay format | Scientific Literature | ||
| 14. | ALA3129772 | B | Competitive inhibition of mouse FAAH preincubated for 6 hrs followed by FP-rhodamine addition measured after 10 mins by fluorescence scanning | Mus musculus | 6 | single protein format | Scientific Literature | ||
| 15. | ALA3129773 | B | Competitive inhibition of mouse heart membrane TGH preincubated for 6 hrs followed by FP-rhodamine addition measured after 10 mins by fluorescence scanning | Mus musculus | 6 | assay format | Scientific Literature | ||
| 16. | ALA3129774 | B | Competitive inhibition of mouse brain membrane KIAA1363 preincubated for 6 hrs followed by FP-rhodamine addition measured after 10 mins by fluorescence scanning | Mus musculus | 6 | assay format | Scientific Literature | ||
| 17. | ALA3129775 | B | Competitive inhibition of mouse brain membrane MAGL preincubated for 6 hrs followed by FP-rhodamine addition measured after 10 mins by fluorescence scanning | Mus musculus | 6 | assay format | Scientific Literature | ||
| 18. | ALA3129917 | B | Noncompetitive inhibition of recombinant rat FAAH expressed in Escherichia coli assessed as breakdown of [14C]-oleamide at 1 to 5 nM preincubated for 3 hrs by Lineweaver-Burk plot analysis | Rattus norvegicus | 2 | assay format | Scientific Literature | ||
| 19. | ALA3129923 | B | Time-dependent inhibition of recombinant rat FAAH expressed in Escherichia coli assessed as breakdown of [14C]-oleamide preincubated for 6 hrs by Dixon plot analysis | Rattus norvegicus | 16 | assay format | Scientific Literature | ||
| 20. | ALA3129924 | B | Time-dependent inhibition of recombinant rat FAAH expressed in Escherichia coli assessed as breakdown of [14C]-oleamide preincubated for 3 hrs by Dixon plot analysis | Rattus norvegicus | 19 | assay format | Scientific Literature |
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