| # | Aladdin ID | Assay Type | Description | Organism | Compounds | Reference | BAO Format | Source | |
|---|---|---|---|---|---|---|---|---|---|
| 1. | ALA3367859 | Binding | Inhibition of TASK-1 (unknown origin) expressed in CHO cells at 3 uM by thallium flux assay | Homo sapiens | 56 | ALA3351482 | cell-based format | Scientific Literature | |
| 2. | ALA3367860 | Binding | Inhibition of TASK-1 (unknown origin) expressed in CHO cells by thallium flux assay | Homo sapiens | 58 | ALA3351482 | cell-based format | Scientific Literature | |
| 3. | ALA3367861 | Binding | Inhibition of TASK-3 (unknown origin) expressed in CHO cells by thallium flux assay | Homo sapiens | 56 | ALA3351482 | cell-based format | Scientific Literature | |
| 4. | ALA3367862 | Binding | Selectivity ratio of IC50 for TASK-3 (unknown origin) to IC50 for TASK-1 (unknown origin) | Homo sapiens | 52 | ALA3351482 | assay format | Scientific Literature | |
| 5. | ALA3367863 | Binding | Inhibition of KCNQ2 (unknown origin) | Homo sapiens | 6 | ALA3351482 | single protein format | Scientific Literature | |
| 6. | ALA3367864 | Binding | Inhibition of human ERG | Homo sapiens | 6 | ALA3351482 | single protein format | Scientific Literature | |
| 7. | ALA3367865 | Binding | Inhibition of Kir2.1 (unknown origin) | Homo sapiens | 5 | ALA3351482 | single protein format | Scientific Literature | |
| 8. | ALA3367868 | Binding | Inhibition of TASK-1 (unknown origin) expressed in CHO cells by QPatch assay | Homo sapiens | 8 | ALA3351482 | cell-based format | Scientific Literature | |
| 9. | ALA3367869 | Binding | Inhibition of TASK-3 (unknown origin) expressed in HEK293 cells by QPatch assay | Homo sapiens | 8 | ALA3351482 | cell-based format | Scientific Literature | |
| 10. | ALA3367870 | Binding | Selectivity ratio of IC50 for TASK-3 (unknown origin) to IC50 for TASK-1 (unknown origin) by QPatch assay | Homo sapiens | 8 | ALA3351482 | assay format | Scientific Literature | |
| 11. | ALA3367871 | Physicochemical | Kinetic solubility of the compound in pION buffer at pH 0 | 5 | ALA3351482 | small-molecule physicochemical format | Scientific Literature | ||
| 12. | ALA3367872 | Physicochemical | Kinetic solubility of the compound in pION buffer at pH 6.2 | 5 | ALA3351482 | small-molecule physicochemical format | Scientific Literature | ||
| 13. | ALA3367873 | Physicochemical | Kinetic solubility of the compound in pION buffer at pH 7.4 | 5 | ALA3351482 | small-molecule physicochemical format | Scientific Literature | ||
| 14. | ALA3367874 | Physicochemical | Kinetic solubility of the compound in PBS buffer at pH 7.4 after 48 hrs by reverse phase HPLC/UV/HRMS system | 5 | ALA3351482 | small-molecule physicochemical format | Scientific Literature | ||
| 15. | ALA3215093 | Functional | PubChem BioAssay. SAR analysis for the identification of selective inhibitors of the two-pore domain potassium channel TASK1(KCNK3):Automated Electrophysiology. (Class of assay: confirmatory) | 17 | ALA1201862 | assay format | PubChem BioAssays | ||
| 16. | ALA3215269 | Functional | PubChem BioAssay. SAR Analysis for the identification of inhibitors of the two-pore domain potassium channel TASK1 (KCNK3). (Class of assay: confirmatory) | 94 | ALA1201862 | assay format | PubChem BioAssays | ||
| 17. | ALA3214982 | Functional | PubChem BioAssay. SAR analysis for the identification of selective inhibitors of the two-pore domain potassium channel TASK1(KCNK3) -selectivity assay against TASK3(KCNK9): Automated Electrophysiology. (Class of assay: confirmatory) | 13 | ALA1201862 | assay format | PubChem BioAssays |
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