# | Aladdin ID | Assay Type | Description | Organism | Compounds | Reference | BAO Format | Source | |
---|---|---|---|---|---|---|---|---|---|
1. | ALA3239420 | F | Agonist activity at human TGR5 expressed in Jurkat cells assessed as intracellular cAMP level after 1 hr by HTRF assay | Homo sapiens | 42 | ALA3232835 | cell-based format | Scientific Literature | |
2. | ALA3239421 | F | Agonist activity at mouse TGR5 expressed in Jurkat cells assessed as intracellular cAMP level after 1 hr by HTRF assay | Mus musculus | 42 | ALA3232835 | cell-based format | Scientific Literature | |
3. | ALA3239423 | A | Inhibition of CYP3A4 (unknown origin) | Homo sapiens | 17 | ALA3232835 | single protein format | Scientific Literature | |
4. | ALA3239424 | B | Inhibition of human ERG by patch clamp method | Homo sapiens | 15 | ALA3232835 | assay format | Scientific Literature | |
5. | ALA3239429 | A | Intrinsic clearance in mouse liver microsomes after 60 mins by HPLC analysis | Mus musculus | 11 | ALA3232835 | assay format | Scientific Literature | |
6. | ALA3239494 | F | Agonist activity at human TGR5 expressed in Jurkat cells assessed as intracellular cAMP level after 1 hr by HTRF assay relative to control | Homo sapiens | 42 | ALA3232835 | cell-based format | Scientific Literature | |
7. | ALA3239495 | F | Agonist activity at mouse TGR5 expressed in Jurkat cells assessed as intracellular cAMP level after 1 hr by HTRF assay relative to control | Mus musculus | 42 | ALA3232835 | cell-based format | Scientific Literature |