| # | Aladdin ID | Assay Type | Description | Organism | Compounds | Reference | BAO Format | Source | |
|---|---|---|---|---|---|---|---|---|---|
| 1. | ALA3268497 | B | Displacement of [9-methyl-3H]BRL-43694 from human 5-HT3A receptor after overnight incubation by scintillation proximity assay | Homo sapiens | 11 | ALA3259590 | single protein format | Scientific Literature | |
| 2. | ALA3268498 | B | Partial agonist activity at human 5-HT3A receptor expressed in HEK293 cells assessed as change in Ca2+ level measured as intrinsic activity at 1 uM relative to 5-HT in presence of carbachol | Homo sapiens | 6 | ALA3259590 | cell-based format | Scientific Literature | |
| 3. | ALA3268499 | B | Partial agonist activity at mouse 5-HT3A receptor expressed in HEK293 cells assessed as change in Ca2+ level measured as intrinsic activity at 1 uM relative to 5-HT in presence of carbachol | Mus musculus | 4 | ALA3259590 | cell-based format | Scientific Literature | |
| 4. | ALA3268500 | B | Agonist activity at human 5-HT3A receptor expressed in HEK293 cells in presence of carbachol | Homo sapiens | 6 | ALA3259590 | cell-based format | Scientific Literature | |
| 5. | ALA3268501 | B | Agonist activity at mouse 5-HT3A receptor expressed in HEK293 cells in presence of carbachol | Mus musculus | 4 | ALA3259590 | cell-based format | Scientific Literature | |
| 6. | ALA3268502 | A | Inhibition of CYP1A2 (unknown origin) | Homo sapiens | 7 | ALA3259590 | single protein format | Scientific Literature | |
| 7. | ALA3268503 | A | Inhibition of CYP2B6 (unknown origin) | Homo sapiens | 6 | ALA3259590 | single protein format | Scientific Literature | |
| 8. | ALA3268874 | A | Inhibition of CYP2C9 (unknown origin) | Homo sapiens | 6 | ALA3259590 | single protein format | Scientific Literature | |
| 9. | ALA3268875 | A | Inhibition of CYP2C19 (unknown origin) | Homo sapiens | 6 | ALA3259590 | single protein format | Scientific Literature | |
| 10. | ALA3268876 | A | Inhibition of CYP2D6 (unknown origin) | Homo sapiens | 6 | ALA3259590 | single protein format | Scientific Literature | |
| 11. | ALA3268877 | A | Inhibition of CYP3A4 (unknown origin) | Homo sapiens | 7 | ALA3259590 | single protein format | Scientific Literature | |
| 12. | ALA3268878 | A | Intrinsic clearance in human liver microsomes | Homo sapiens | 8 | ALA3259590 | assay format | Scientific Literature |
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