| # | Aladdin ID | Assay Type | Description | Organism | Compounds | Reference | BAO Format | Source | |
|---|---|---|---|---|---|---|---|---|---|
| 1. | ALA3270094 | F | Agonist activity at human beta-2 adrenergic receptor expressed in human H292 cells assessed as accumulation of intracellular cAMP after 1 hr by AlphaScreen assay | Homo sapiens | 17 | ALA3259656 | cell-based format | Scientific Literature | |
| 2. | ALA3270095 | B | Intrinsic activity at human beta-2 adrenergic receptor expressed in human H292 cells relative to formoterol | Homo sapiens | 17 | ALA3259656 | cell-based format | Scientific Literature | |
| 3. | ALA3270096 | B | Selectivity ratio of IC50 for human recombinant beta-1 adrenergic receptor expressed in CHO cells to IC50 for human beta-2 adrenergic receptor expressed in human H292 cells | Homo sapiens | 1 | ALA3259656 | cell-based format | Scientific Literature | |
| 4. | ALA3270097 | B | Selectivity ratio of IC50 for human beta-3 adrenergic receptor to IC50 for human beta-2 adrenergic receptor expressed in human H292 cells | Homo sapiens | 1 | ALA3259656 | cell-based format | Scientific Literature | |
| 5. | ALA3270098 | B | Selectivity ratio of IC50 for human recombinant dopamine D2S receptor expressed in HEK cells to IC50 for human beta-2 adrenergic receptor expressed in human H292 cells | Homo sapiens | 1 | ALA3259656 | cell-based format | Scientific Literature | |
| 6. | ALA3270099 | B | Selectivity ratio of IC50 for human recombinant alpha-1D adrenergic receptor expressed in HEK cells to IC50 for human beta-2 adrenergic receptor expressed in human H292 cells | Homo sapiens | 1 | ALA3259656 | cell-based format | Scientific Literature | |
| 7. | ALA3270100 | F | Agonist activity at human recombinant alpha-1D adrenergic receptor expressed in HEK cells assessed as accumulation of intracellular cAMP | Homo sapiens | 1 | ALA3259656 | cell-based format | Scientific Literature | |
| 8. | ALA3270101 | B | Selectivity ratio of EC50 for human recombinant dopamine D2S receptor expressed in HEK cells to EC50 for human beta-2 adrenergic receptor expressed in human H292 cells | Homo sapiens | 1 | ALA3259656 | cell-based format | Scientific Literature | |
| 9. | ALA3270481 | F | Partial agonist activity at human recombinant dopamine D2S receptor expressed in HEK cells by GTPgammaS binding assay | Homo sapiens | 1 | ALA3259656 | cell-based format | Scientific Literature | |
| 10. | ALA3270483 | F | Agonist activity at human recombinant beta-1 adrenergic receptor expressed in CHO cells assessed as accumulation of intracellular cAMP | Homo sapiens | 4 | ALA3259656 | cell-based format | Scientific Literature | |
| 11. | ALA3270484 | B | Intrinsic activity at beta-2 adrenergic receptor in guinea pig tracheal rings | Cavia porcellus | 5 | ALA3259656 | single protein format | Scientific Literature | |
| 12. | ALA3270485 | B | Agonist activity at beta-2 adrenergic receptor in human bronchial rings assessed as time required to reach 90% of final relaxation of carbachol-constricted bronchial rings | Homo sapiens | 9 | ALA3259656 | single protein format | Scientific Literature | |
| 13. | ALA3270486 | B | Agonist activity at beta-2 adrenergic receptor in guinea pig tracheal rings assessed as time required to reach 90% of final relaxation of methacholine-constricted tracheal rings | Cavia porcellus | 10 | ALA3259656 | single protein format | Scientific Literature | |
| 14. | ALA3270487 | B | Agonist activity at beta-2 adrenergic receptor in guinea pig tracheal rings assessed as relaxation of methacholine-constricted tracheal rings | Cavia porcellus | 5 | ALA3259656 | single protein format | Scientific Literature | |
| 15. | ALA3270488 | F | Agonist activity at beta-2 adrenergic receptor in rat C6 cells assessed as cAMP accumulation | Rattus norvegicus | 1 | ALA3259656 | cell-based format | Scientific Literature | |
| 16. | ALA3270489 | B | Intrinsic activity at beta-2 adrenergic receptor in rat C6 cells | Rattus norvegicus | 1 | ALA3259656 | cell-based format | Scientific Literature | |
| 17. | ALA3270490 | B | Agonist activity at rabbit recombinant beta-2 adrenergic receptor assessed as cAMP accumulation by cell-based assay | Oryctolagus cuniculus | 1 | ALA3259656 | cell-based format | Scientific Literature | |
| 18. | ALA3270491 | F | Agonist activity at dog recombinant beta-2 adrenergic receptor assessed as cAMP accumulation by cell-based assay | Canis lupus familiaris | 1 | ALA3259656 | cell-based format | Scientific Literature | |
| 19. | ALA3270492 | B | Intrinsic activity at dog recombinant beta-2 adrenergic receptor | Canis lupus familiaris | 1 | ALA3259656 | single protein format | Scientific Literature | |
| 20. | ALA3270493 | F | Agonist activity at mouse recombinant beta-2 adrenergic receptor assessed as cAMP accumulation by cell-based assay | Mus musculus | 1 | ALA3259656 | cell-based format | Scientific Literature |
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