Inhibition of human placental 17beta-HSD1 cytosolic fraction using [2, 4, 6, 7-3H]-estrone as substrate at 1 uM after 10 mins by HPLC analysis relative to control
Inhibition of human placental 17beta-HSD2 microsomal fraction using [2, 4, 6, 7-3H]-estradiol as substrate at 1 uM after 20 mins by HPLC analysis relative to control
Inhibition of recombinant mouse 17beta-HSD1 expressed in HEK293 cells using [3H]-estrone as substrate at 1 uM after 10 mins by HPLC analysis relative to control