| # | Aladdin ID | Assay Type | Description | Organism | Compounds | Reference | BAO Format | Source | |
|---|---|---|---|---|---|---|---|---|---|
| 1. | ALA3368107 | P | Octanol-water partition coefficient, log D of the compound at pH 7.4 by shake flask method | 14 | ALA3352699 | small-molecule physicochemical format | Scientific Literature | ||
| 2. | ALA3368108 | B | Inhibition of human GPR103 receptor expressed in CHOK1 cells by IP-1 assay | Homo sapiens | 14 | ALA3352699 | cell-based format | Scientific Literature | |
| 3. | ALA3368109 | B | Displacement of [125I]QRFP43 from human GPR103 receptor expressed in HEK cells after 90 mins incubation by scintillation counting | Homo sapiens | 3 | ALA3352699 | cell-based format | Scientific Literature | |
| 4. | ALA3368110 | B | Inhibition of mouse GPR103A receptor expressed in CHO cells by IP-1 assay | Mus musculus | 3 | ALA3352699 | cell-based format | Scientific Literature | |
| 5. | ALA3368352 | B | Inhibition of mouse GPR103B receptor expressed in CHO cells by IP-1 assay | Mus musculus | 3 | ALA3352699 | cell-based format | Scientific Literature | |
| 6. | ALA3368353 | P | Solubility of the compound in HBSS buffer at pH 7.4 after 18 hrs by LC/MS/MS analysis | 3 | ALA3352699 | small-molecule physicochemical format | Scientific Literature | ||
| 7. | ALA3368354 | A | Intrinsic clearance in human hepatocytes measured per 10'6 cells | Homo sapiens | 3 | ALA3352699 | cell-based format | Scientific Literature | |
| 8. | ALA3368355 | A | Intrinsic clearance in human liver microsomes | Homo sapiens | 3 | ALA3352699 | assay format | Scientific Literature | |
| 9. | ALA3368356 | A | Apparent permeability across apical to basolateral side in human Caco2 cells by LC-MS/MS analysis | Homo sapiens | 3 | ALA3352699 | cell-based format | Scientific Literature | |
| 10. | ALA3368357 | A | Inhibition of human CYP2D6 after 20 to 50 mins by high-throughput fluorescence assay | Homo sapiens | 3 | ALA3352699 | single protein format | Scientific Literature | |
| 11. | ALA3368358 | B | Inhibition of human ERG expressed in CHO cells by electrophysiology assay | Homo sapiens | 3 | ALA3352699 | cell-based format | Scientific Literature | |
| 12. | ALA3368359 | B | Inhibition of human Nav1.5 expressed in CHO cells by electrophysiology assay | Homo sapiens | 3 | ALA3352699 | cell-based format | Scientific Literature | |
| 13. | ALA3368360 | B | Inhibition of human cardiac slowly activating delayed rectifier K+ channel expressed in CHO cells by electrophysiology assay | Homo sapiens | 3 | ALA3352699 | cell-based format | Scientific Literature | |
| 14. | ALA3368361 | A | Inhibition of human recombinant CYP3A4 after 20 to 50 mins by high-throughput fluorescence assay | Homo sapiens | 2 | ALA3352699 | single protein format | Scientific Literature | |
| 15. | ALA3368362 | A | Inhibition of human recombinant CYP1A2 after 20 to 50 mins by high-throughput fluorescence assay | Homo sapiens | 2 | ALA3352699 | single protein format | Scientific Literature | |
| 16. | ALA3368363 | A | Inhibition of human recombinant CYP2C8 after 20 to 50 mins by high-throughput fluorescence assay | Homo sapiens | 2 | ALA3352699 | single protein format | Scientific Literature | |
| 17. | ALA3368364 | A | Inhibition of human recombinant CYP2C9 after 20 to 50 mins by high-throughput fluorescence assay | Homo sapiens | 2 | ALA3352699 | single protein format | Scientific Literature | |
| 18. | ALA3368365 | A | Inhibition of human recombinant CYP2C19 after 20 to 50 mins by high-throughput fluorescence assay | Homo sapiens | 2 | ALA3352699 | single protein format | Scientific Literature | |
| 19. | ALA3368370 | B | Selectivity index, ratio of IC50 for mouse GPR103A receptor to IC50 for mouse GPR103B receptor | Mus musculus | 2 | ALA3352699 | assay format | Scientific Literature |
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