| # | Aladdin ID | Assay Type | Description | Organism | Compounds | Reference | BAO Format | Source | |
|---|---|---|---|---|---|---|---|---|---|
| 1. | ALA3368976 | B | Inhibition of human recombinant GST-tagged PDE10A using [3H]-cAMP as substrate at 1 uM after 30 mins by scintillation proximity assay | Homo sapiens | 18 | ALA3352660 | single protein format | Scientific Literature | |
| 2. | ALA3368977 | B | Inhibition of human recombinant GST-tagged PDE10A using [3H]-cAMP as substrate after 30 mins by scintillation proximity assay | Homo sapiens | 18 | ALA3352660 | single protein format | Scientific Literature | |
| 3. | ALA3368978 | B | Inhibition of rat recombinant GST-tagged PDE10A using [3H]-cAMP as substrate by scintillation proximity assay | Rattus norvegicus | 14 | ALA3352660 | single protein format | Scientific Literature | |
| 4. | ALA3368979 | B | Inhibition of mouse recombinant GST-tagged PDE10A using [3H]-cAMP as substrate after 30 mins by scintillation proximity assay | Mus musculus | 5 | ALA3352660 | single protein format | Scientific Literature | |
| 5. | ALA3368980 | B | Inhibition of human recombinant PDE2A using cAMP as substrate at 1 uM after 30 mins by HTRF method | Homo sapiens | 10 | ALA3352660 | single protein format | Scientific Literature | |
| 6. | ALA3368981 | B | Inhibition of human recombinant PDE2A using cAMP as substrate at 10 uM after 30 mins by HTRF method | Homo sapiens | 10 | ALA3352660 | single protein format | Scientific Literature | |
| 7. | ALA3368982 | B | Inhibition of human recombinant PDE3A using cAMP as substrate at 1 uM after 30 mins by HTRF method | Homo sapiens | 10 | ALA3352660 | single protein format | Scientific Literature | |
| 8. | ALA3368983 | B | Inhibition of human recombinant PDE3A using cAMP as substrate at 10 uM after 30 mins by HTRF method | Homo sapiens | 10 | ALA3352660 | single protein format | Scientific Literature | |
| 9. | ALA3368984 | B | Inhibition of human recombinant PDE4D using [3H]-cAMP as substrate at 1 uM after 30 mins by two-step radiometric assay | Homo sapiens | 10 | ALA3352660 | single protein format | Scientific Literature | |
| 10. | ALA3368985 | B | Inhibition of human recombinant PDE4D using [3H]-cAMP as substrate at 10 uM after 30 mins by two-step radiometric assay | Homo sapiens | 10 | ALA3352660 | single protein format | Scientific Literature | |
| 11. | ALA3368986 | B | Inhibition of human recombinant PDE5A using [3H]-cAMP as substrate at 1 uM after 30 mins by scintillation proximity assay | Homo sapiens | 10 | ALA3352660 | single protein format | Scientific Literature | |
| 12. | ALA3368987 | B | Inhibition of human recombinant PDE5A using [3H]-cAMP as substrate at 10 uM after 30 mins by scintillation proximity assay | Homo sapiens | 10 | ALA3352660 | single protein format | Scientific Literature | |
| 13. | ALA3368988 | B | Inhibition of human recombinant PDE7A using [3H]-cAMP as substrate at 1 uM after 30 mins by two-step radiometric assay | Homo sapiens | 10 | ALA3352660 | single protein format | Scientific Literature | |
| 14. | ALA3368989 | B | Inhibition of human recombinant PDE7A using [3H]-cAMP as substrate at 10 uM after 30 mins by two-step radiometric assay | Homo sapiens | 10 | ALA3352660 | single protein format | Scientific Literature | |
| 15. | ALA3368990 | B | Inhibition of human recombinant PDE11A using [3H]-cAMP as substrate at 1 uM after 30 mins by two-step radiometric assay | Homo sapiens | 10 | ALA3352660 | single protein format | Scientific Literature | |
| 16. | ALA3368991 | B | Inhibition of human recombinant PDE11A using [3H]-cAMP as substrate at 10 uM after 30 mins by two-step radiometric assay | Homo sapiens | 10 | ALA3352660 | single protein format | Scientific Literature | |
| 17. | ALA3368992 | A | Metabolic stability in Wistar rat liver microsomes incubated for 10 mins prior to NADPH addition measured after 60 mins by LC/MS/MS analysis | Rattus norvegicus | 12 | ALA3352660 | assay format | Scientific Literature | |
| 18. | ALA3368993 | A | Metabolic stability in CD1 mouse liver microsomes incubated for 10 mins prior to NADPH addition measured after 60 mins by LC/MS/MS analysis | Mus musculus | 12 | ALA3352660 | assay format | Scientific Literature | |
| 19. | ALA3368994 | A | Metabolic stability in Beagle dog liver microsomes incubated for 10 mins prior to NADPH addition measured after 60 mins by LC/MS/MS analysis | Canis lupus familiaris | 12 | ALA3352660 | assay format | Scientific Literature | |
| 20. | ALA3368995 | A | Metabolic stability in cynomolgus monkey liver microsomes incubated for 10 mins prior to NADPH addition measured after 60 mins by LC/MS/MS analysis | Macaca fascicularis | 12 | ALA3352660 | assay format | Scientific Literature |
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