| # | Aladdin ID | Assay Type | Description | Organism | Compounds | Reference | BAO Format | Source | |
|---|---|---|---|---|---|---|---|---|---|
| 1. | ALA3371410 | P | Retention time of the compound measured over 15 mins at flow rate of 0.5 mL/min by HPLC | 18 | small-molecule physicochemical format | Scientific Literature | |||
| 2. | ALA3371411 | P | Retention time of the compound measured over 30 mins at flow rate of 1 mL/min by HPLC | 21 | small-molecule physicochemical format | Scientific Literature | |||
| 3. | ALA3371413 | B | Inhibition of human Nav1.7 expressed in HEK-293 cells at -130 to -110 mV holding potential by whole-cell voltage clamp analysis | Homo sapiens | 21 | cell-based format | Scientific Literature | ||
| 4. | ALA3371414 | B | Inhibition of rat Nav1.7 expressed in HEK-293 cells at -130 to -110 mV holding potential by whole-cell voltage clamp analysis | Rattus norvegicus | 21 | cell-based format | Scientific Literature | ||
| 5. | ALA3371415 | B | Selectivity ratio of IC50 for rat Nav1.2 expressed in HEK-293 cells to IC50 for human Nav1.7 expressed in HEK-293 cells | 18 | cell-based format | Scientific Literature | |||
| 6. | ALA3371419 | B | Inhibition of human Nav1.7 expressed in HEK-293 cells assessed as time for channel-mediated current inhibition at 3 nM by time-course experiment | Homo sapiens | 1 | cell-based format | Scientific Literature | ||
| 7. | ALA3419342 | B | Inhibition of human NaV1.7 at -140 mV holding potential by whole-cell patch clamp assay | Homo sapiens | 70 | assay format | Scientific Literature | ||
| 8. | ALA3419343 | B | Inhibition of human NaV1.5 at -140 mV holding potential by whole-cell patch clamp assay | Homo sapiens | 70 | assay format | Scientific Literature | ||
| 9. | ALA3419344 | B | Inhibition of human NaV1.4 at -140 mV holding potential by whole-cell patch clamp assay | Homo sapiens | 70 | assay format | Scientific Literature | ||
| 10. | ALA4266772 | B | Inhibition of human Nav1.7 expressed in HEK293 cells at holding potential of -120 mV by manual electrophysiology method | Homo sapiens | 1 | cell-based format | Scientific Literature | ||
| 11. | ALA4266773 | B | Selectivity index, ratio of IC50 for human Nav1.1 to IC50 for human Nav1.7 | Homo sapiens | 1 | assay format | Scientific Literature | ||
| 12. | ALA4266774 | B | Selectivity index, ratio of IC50 for human Nav1.2 to IC50 for human Nav1.7 | Homo sapiens | 1 | assay format | Scientific Literature | ||
| 13. | ALA4266775 | B | Selectivity index, ratio of IC50 for human Nav1.3 to IC50 for human Nav1.7 | Homo sapiens | 1 | assay format | Scientific Literature | ||
| 14. | ALA4266776 | B | Selectivity index, ratio of IC50 for human Nav1.4 to IC50 for human Nav1.7 | Homo sapiens | 1 | assay format | Scientific Literature | ||
| 15. | ALA4266777 | B | Selectivity index, ratio of IC50 for human Nav1.5 to IC50 for human Nav1.7 | Homo sapiens | 1 | assay format | Scientific Literature | ||
| 16. | ALA4266778 | B | Selectivity index, ratio of IC50 for human Nav1.6 to IC50 for human Nav1.7 | Homo sapiens | 1 | assay format | Scientific Literature | ||
| 17. | ALA4321987 | B | Inhibition of human Nav1.7 expressed in HEK293 cells by electrophysiology assay | Homo sapiens | 15 | cell-based format | Scientific Literature | ||
| 18. | ALA4321991 | B | Inhibition of human Nav1.1 expressed in HEK293 cells by electrophysiology assay | Homo sapiens | 11 | cell-based format | Scientific Literature | ||
| 19. | ALA4321992 | B | Inhibition of human Nav1.2 expressed in HEK293 cells by electrophysiology assay | Homo sapiens | 12 | cell-based format | Scientific Literature | ||
| 20. | ALA4321993 | B | Inhibition of human Nav1.3 expressed in HEK293 cells by electrophysiology assay | Homo sapiens | 8 | cell-based format | Scientific Literature |
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