| # | Aladdin ID | Assay Type | Description | Organism | Compounds | Reference | BAO Format | Source | |
|---|---|---|---|---|---|---|---|---|---|
| 1. | ALA3364949 | Binding | Inhibition of fluorescein-labeled human GK interaction with biotin-labeled human GKRP compound incubated for 20 mins prior to addition of fluorescein-labeled GK measured after 2 to 4 hrs by AlphaScreen assay | Homo sapiens | 45 | ALA3352455 | single protein format | Scientific Literature | |
| 2. | ALA3364950 | Binding | Induction of GK translocation from nucleus to cytoplasm of mouse hepatocytes preincubated for 20 mins followed by glucose challenge measured after 40 mins by Hoechst 33342 staining-based assay | Mus musculus | 40 | ALA3352455 | cell-based format | Scientific Literature | |
| 3. | ALA3364951 | ADME | Intrinsic clearance in human liver microsomes at 1 uM after 30 mins in presence of NADPH | Homo sapiens | 45 | ALA3352455 | assay format | Scientific Literature | |
| 4. | ALA3364952 | ADME | Intrinsic clearance in rat liver microsomes at 1 uM after 30 mins in presence of NADPH | Rattus norvegicus | 45 | ALA3352455 | assay format | Scientific Literature |
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