| # | Aladdin ID | Assay Type | Description | Organism | Compounds | Reference | BAO Format | Source | |
|---|---|---|---|---|---|---|---|---|---|
| 1. | ALA3371274 | B | Inhibition of proteasome subunit beta-1i in human Raji cells using BODIPY- epoxomicin by fluorescent densitometry | Homo sapiens | 21 | cell-based format | Scientific Literature | ||
| 2. | ALA3371275 | B | Inhibition of 20s proteasome subunit beta-1c in human Raji cells using BODIPY- epoxomicin by fluorescent densitometry | Homo sapiens | 21 | cell-based format | Scientific Literature | ||
| 3. | ALA3371276 | B | Inhibition of proteasome subunit beta-2i in human Raji cells using BODIPY- epoxomicin by fluorescent densitometry | Homo sapiens | 13 | cell-based format | Scientific Literature | ||
| 4. | ALA3371278 | B | Ratio of IC50 for proteasome subunit beta-1i to IC50 for proteasome subunit beta-5i in human Raji cells | Homo sapiens | 13 | cell-based format | Scientific Literature | ||
| 5. | ALA3371291 | B | Ratio of IC50 for 20s proteasome subunit beta-1c to IC50 for proteasome subunit beta-1i in human Raji cells | Homo sapiens | 13 | cell-based format | Scientific Literature | ||
| 6. | ALA4394491 | B | Inhibition of purified human 20S immunoproteasome beta1 subunit using Ac-Pro-Ala-Leu-AMC as substrate pretreated for 1 hr followed by substrate addition and measured at 1 min interval by fluorescence assay | Homo sapiens | 4 | single protein format | Scientific Literature | ||
| 7. | ALA4394492 | F | Cytotoxicity against human NCI-H23 cells after 72 hrs by CellTiter 96 AQueous one solution cell proliferation assay | Homo sapiens | 10 | cell-based format | Scientific Literature | ||
| 8. | ALA4394493 | F | Cytotoxicity against human NCI-H727 cells after 72 hrs by CellTiter 96 AQueous one solution cell proliferation assay | Homo sapiens | 10 | cell-based format | Scientific Literature | ||
| 9. | ALA4394494 | F | Selectivity ratio of IC50 for human NCI-H727 cells to IC50 for human NCI-H23 cells | Homo sapiens | 6 | assay format | Scientific Literature | ||
| 10. | ALA4394495 | F | Cytotoxicity against human RPMI8226 cells after 72 hrs by CellTiter 96 AQueous one solution cell proliferation assay | Homo sapiens | 4 | cell-based format | Scientific Literature | ||
| 11. | ALA4394496 | F | Cytotoxicity against human RPMI8226/Cfzr cells after 72 hrs by CellTiter 96 AQueous one solution cell proliferation assay | Homo sapiens | 6 | cell-based format | Scientific Literature | ||
| 12. | ALA4394497 | F | Selectivity ratio of IC50 for human RPMI8226/Cfzr cells to IC50 for human RPMI8226 cells | Homo sapiens | 4 | assay format | Scientific Literature | ||
| 13. | ALA4394500 | F | Cytotoxicity against human multiple myeloma cells at 10 uM after 48 hrs by CellTiter 96 AQueous one solution cell proliferation assay | Homo sapiens | 2 | cell-based format | Scientific Literature | ||
| 14. | ALA4394501 | F | Cytotoxicity against human Btz-resistant multiple myeloma cells at 10 uM after 48 hrs by CellTiter 96 AQueous one solution cell proliferation assay | Homo sapiens | 2 | cell-based format | Scientific Literature | ||
| 15. | ALA4394502 | B | Inhibition of 20S proteasome beta5 subunit in human RPMI8226 cell lysate using Suc-LLVY-AMC as substrate pretreated for 1 hr followed by substrate addition and measured at 1 min interval by fluorescence assay | Homo sapiens | 9 | subcellular format | Scientific Literature |
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