| # | Aladdin ID | Assay Type | Description | Organism | Compounds | Reference | BAO Format | Source | |
|---|---|---|---|---|---|---|---|---|---|
| 1. | ALA3378627 | T | Toxicity in anesthetized vagus-intact cardiovascular dog model assessed as QTc interval prolongation at 909 uM plasma concentration | Canis lupus familiaris | 1 | ALA3352784 | organism-based format | Scientific Literature | |
| 2. | ALA3378631 | A | Cmax in anesthetized vagus-intact cardiovascular dog model at 10 mg/kg, iv for 30 mins | Canis lupus familiaris | 2 | ALA3352784 | organism-based format | Scientific Literature | |
| 3. | ALA3378632 | A | Cmax in anesthetized vagus-intact cardiovascular dog model at 20 mg/kg, iv for 30 mins | Canis lupus familiaris | 2 | ALA3352784 | organism-based format | Scientific Literature | |
| 4. | ALA3378633 | A | Cmax in anesthetized vagus-intact cardiovascular dog model at 30 mg/kg, iv for 30 mins | Canis lupus familiaris | 2 | ALA3352784 | organism-based format | Scientific Literature | |
| 5. | ALA3378637 | B | Inhibition of human ERG by MK-499 displacement binding analysis | Homo sapiens | 12 | ALA3352784 | single protein format | Scientific Literature | |
| 6. | ALA3378639 | B | Displacement of [125I]SS-14 from human SSTR3 expressed in CHO cells by TopCount analyzer | Homo sapiens | 16 | ALA3352784 | cell-based format | Scientific Literature | |
| 7. | ALA3378640 | F | Antagonist activity at human SSTR3 expressed in CHO cells assessed as cAMP level by fluorescence analysis | Homo sapiens | 16 | ALA3352784 | cell-based format | Scientific Literature | |
| 8. | ALA3378641 | B | Displacement of [125I]SS-14 from mouse SSTR3 expressed in CHO cells by TopCount analyzer | Mus musculus | 16 | ALA3352784 | cell-based format | Scientific Literature | |
| 9. | ALA3378642 | F | Antagonist activity at mouse SSTR3 expressed in CHO cells assessed as cAMP level by fluorescence analysis | Mus musculus | 16 | ALA3352784 | cell-based format | Scientific Literature | |
| 10. | ALA3378643 | F | Antagonist activity at human SSTR3 expressed in CHO cells assessed as cAMP level by fluorescence analysis relative to control | Homo sapiens | 16 | ALA3352784 | cell-based format | Scientific Literature | |
| 11. | ALA3378644 | F | Antagonist activity at mouse SSTR3 expressed in CHO cells assessed as cAMP level by fluorescence analysis relative to control | Mus musculus | 16 | ALA3352784 | cell-based format | Scientific Literature | |
| 12. | ALA3378646 | B | Inhibition of human ERG at 30 uM by functional patch clamp assay | Homo sapiens | 2 | ALA3352784 | assay format | Scientific Literature | |
| 13. | ALA3378647 | A | Clearance in mouse | Mus musculus | 1 | ALA3352784 | organism-based format | Scientific Literature | |
| 14. | ALA3378648 | A | Half life in mouse | Mus musculus | 1 | ALA3352784 | organism-based format | Scientific Literature | |
| 15. | ALA3378649 | A | Oral bioavailability in mouse | Mus musculus | 1 | ALA3352784 | organism-based format | Scientific Literature | |
| 16. | ALA3378650 | B | Displacement of [125I]SS-14 from human SSTR1 expressed in CHO cells by TopCount analyzer | Homo sapiens | 1 | ALA3352784 | cell-based format | Scientific Literature | |
| 17. | ALA3378651 | B | Displacement of [125I]SS-14 from human SSTR2 expressed in CHO cells by TopCount analyzer | Homo sapiens | 1 | ALA3352784 | cell-based format | Scientific Literature | |
| 18. | ALA3378652 | B | Displacement of [125I]SS-14 from human SSTR4 expressed in CHO cells by TopCount analyzer | Homo sapiens | 1 | ALA3352784 | cell-based format | Scientific Literature | |
| 19. | ALA3378653 | B | Displacement of [125I]SS-14 from human SSTR5 expressed in CHO cells by TopCount analyzer | Homo sapiens | 1 | ALA3352784 | cell-based format | Scientific Literature | |
| 20. | ALA3378654 | B | Selectivity ratio of IC50 for human SSTR1 to IC50 for human SSTR3 | Homo sapiens | 1 | ALA3352784 | assay format | Scientific Literature |
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