| # | Aladdin ID | Assay Type | Description | Organism | Compounds | Reference | BAO Format | Source | |
|---|---|---|---|---|---|---|---|---|---|
| 1. | ALA3372166 | B | Displacement of [125I]glucagon from glucagon receptor in rat hepatocyte membranes after 30 mins by gamma-counting | Rattus norvegicus | 21 | cell membrane format | Scientific Literature | ||
| 2. | ALA3372167 | F | Inhibition of glucagon-induced glucagon receptor-mediated cAMP production in rat hepatocytes after 15 mins by cAMP dynamic2 assay | Rattus norvegicus | 1 | cell-based format | Scientific Literature | ||
| 3. | ALA3372168 | B | Inhibition of glucagon-induced glucagon receptor-mediated cAMP production in dog hepatocytes after 15 mins by cAMP dynamic2 assay | Canis lupus familiaris | 1 | cell-based format | Scientific Literature | ||
| 4. | ALA3372712 | F | Inhibition of glucagon-induced glucagon receptor-mediated cAMP production in human hepatocytes after 15 mins by cAMP dynamic2 assay | Homo sapiens | 1 | cell-based format | Scientific Literature | ||
| 5. | ALA3372713 | B | Inhibition of GLP-1R (unknown origin) | Homo sapiens | 1 | single protein format | Scientific Literature | ||
| 6. | ALA3372714 | B | Inhibition of human ERG | Homo sapiens | 1 | single protein format | Scientific Literature | ||
| 7. | ALA3372715 | B | Inhibition of sodium channel site 2 (unknown origin) | Homo sapiens | 1 | assay format | Scientific Literature | ||
| 8. | ALA3372716 | A | Clearance in rat at 1 mg/kg, iv | Rattus norvegicus | 1 | organism-based format | Scientific Literature | ||
| 9. | ALA3372717 | A | Half life in rat at 1 mg/kg, iv | Rattus norvegicus | 1 | organism-based format | Scientific Literature | ||
| 10. | ALA3372718 | A | Volume of distribution at steady state in rat at 1 mg/kg, iv | Rattus norvegicus | 1 | organism-based format | Scientific Literature | ||
| 11. | ALA3372719 | A | Cmax in rat at 1 mg/kg, po | Rattus norvegicus | 1 | organism-based format | Scientific Literature | ||
| 12. | ALA3372720 | A | Half life in rat at 1 mg/kg, po | Rattus norvegicus | 1 | organism-based format | Scientific Literature | ||
| 13. | ALA3372721 | A | Oral bioavailability in rat at 1 mg/kg | Rattus norvegicus | 1 | organism-based format | Scientific Literature | ||
| 14. | ALA3372722 | F | Inhibition of glucagon-induced glucose elevation in rat at 30 mg/kg, po administered 30 mins prior challenge measured up to 6 hrs | Rattus norvegicus | 1 | organism-based format | Scientific Literature | ||
| 15. | ALA3372723 | F | Inhibition of glucagon-induced glucose elevation in non-obese type 2 diabetic Goto-Kakizaki rat at 30 mg/kg, po administered 30 mins prior challenge measured up to 6 hrs | Rattus norvegicus | 1 | organism-based format | Scientific Literature |
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