| # | Aladdin ID | Assay Type | Description | Organism | Compounds | Reference | BAO Format | Source | |
|---|---|---|---|---|---|---|---|---|---|
| 1. | ALA3390270 | B | Inhibition of human PDE2A expressed in Sf9 cells incubated for 40 mins using [3H]-cGMP substrate by scintillation counting method | Homo sapiens | 11 | ALA3351311 | cell-based format | Scientific Literature | |
| 2. | ALA3390271 | B | Inhibition of rat PDE10A expressed in Sf9 cells incubated for 60 mins using [3H]-cAMP substrate by scintillation counting method | Rattus norvegicus | 11 | ALA3351311 | cell-based format | Scientific Literature | |
| 3. | ALA3390272 | B | Selectivity index, ratio of IC50 for rat PDE10A to IC50 for human PDE2A | 11 | ALA3351311 | assay format | Scientific Literature | ||
| 4. | ALA3390273 | B | Selectivity index, ratio of IC50 for human PDE11A to IC50 for human PDE2A | Homo sapiens | 1 | ALA3351311 | assay format | Scientific Literature | |
| 5. | ALA3390274 | B | Inhibition of human PDE1A by scintillation counting method | Homo sapiens | 1 | ALA3351311 | single protein format | Scientific Literature | |
| 6. | ALA3390275 | B | Inhibition of human PDE3B by scintillation counting method | Homo sapiens | 1 | ALA3351311 | single protein format | Scientific Literature | |
| 7. | ALA3390276 | B | Inhibition of human PDE4D by scintillation counting method | Homo sapiens | 1 | ALA3351311 | single protein format | Scientific Literature | |
| 8. | ALA3390277 | B | Inhibition of human PDE5A3 expressed in Sf9 cells by scintillation counting method | Homo sapiens | 1 | ALA3351311 | cell-based format | Scientific Literature | |
| 9. | ALA3390278 | B | Inhibition of human PDE6AB expressed in Sf9 cells by scintillation counting method | Homo sapiens | 1 | ALA3351311 | cell-based format | Scientific Literature | |
| 10. | ALA3390279 | B | Inhibition of human PDE7A1 expressed in Sf9 cells by scintillation counting method | Homo sapiens | 1 | ALA3351311 | cell-based format | Scientific Literature | |
| 11. | ALA3390280 | B | Inhibition of human PDE9A1 expressed in Sf9 cells by scintillation counting method | Homo sapiens | 1 | ALA3351311 | cell-based format | Scientific Literature | |
| 12. | ALA3390281 | B | Inhibition of human PDE11A4 expressed in Sf9 cells by scintillation counting method | Homo sapiens | 1 | ALA3351311 | cell-based format | Scientific Literature | |
| 13. | ALA3381166 | A | Stability in human liver microsomes assessed as parent compound remaining after 15 mins | Homo sapiens | 1 | ALA3351311 | assay format | Scientific Literature | |
| 14. | ALA3381167 | A | Stability in rat liver microsomes assessed as parent compound remaining after 15 mins | Rattus norvegicus | 1 | ALA3351311 | assay format | Scientific Literature | |
| 15. | ALA3381168 | P | Formulatability in water at pH 3.6 | 1 | ALA3351311 | small-molecule physicochemical format | Scientific Literature | ||
| 16. | ALA3381169 | P | Formulatability in 10% beta-HP-CD at pH 3.6 | 1 | ALA3351311 | small-molecule physicochemical format | Scientific Literature | ||
| 17. | ALA3381170 | P | Formulatability in 20% beta-HP-CD at pH 7.0 | 1 | ALA3351311 | small-molecule physicochemical format | Scientific Literature | ||
| 18. | ALA3381171 | A | Inhibition of CYP1A2 in human liver microsomes | Homo sapiens | 1 | ALA3351311 | assay format | Scientific Literature | |
| 19. | ALA3381172 | A | Inhibition of CYP2C9 in human liver microsomes | Homo sapiens | 1 | ALA3351311 | assay format | Scientific Literature | |
| 20. | ALA3381173 | A | Inhibition of CYP2D6 in human liver microsomes | Homo sapiens | 1 | ALA3351311 | assay format | Scientific Literature |
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