# | Aladdin ID | Assay Type | Description | Organism | Compounds | Reference | BAO Format | Source | |
---|---|---|---|---|---|---|---|---|---|
1. | ALA3384537 | Binding | Inhibition of Trypanosoma brucei GSK3 using biotinylated GSP2 substrate by flashplate assay | Trypanosoma brucei | 51 | ALA3352013 | assay format | Scientific Literature | |
2. | ALA3384538 | Binding | Inhibition of human GSK3 using biotinylated GSP2 substrate by flashplate assay | Homo sapiens | 51 | ALA3352013 | protein format | Scientific Literature | |
3. | ALA3385151 | Binding | Selectivity ratio, ratio of IC50 for human GSK3 to IC50 Trypanosoma brucei GSK3 | 51 | ALA3352013 | assay format | Scientific Literature | ||
4. | ALA3385152 | Binding | Inhibition of human CDK2/cyclin A using Biotin-C6-PKTPKKAKKL substrate | Homo sapiens | 51 | ALA3352013 | protein complex format | Scientific Literature | |
5. | ALA3385153 | Binding | Selectivity ratio, ratio of IC50 for human CDK2/cyclin A to IC50 for Trypanosoma brucei GSK3 | 51 | ALA3352013 | assay format | Scientific Literature | ||
6. | ALA3385154 | Functional | Trypanocidal activity against bloodstream stage of Trypanosoma brucei brucei assessed as inhibition of proliferation after 72 hrs | Trypanosoma brucei brucei | 51 | ALA3352013 | organism-based format | Scientific Literature | |
7. | ALA3385155 | ADME | Cytotoxicity against human MRC5 cells assessed as growth inhibition after 72 hrs | Homo sapiens | 51 | ALA3352013 | cell-based format | Scientific Literature |