| # | Aladdin ID | Assay Type | Description | Organism | Compounds | Reference | BAO Format | Source | |
|---|---|---|---|---|---|---|---|---|---|
| 1. | ALA646234 | F | Functional agonism of the compounds to constrict tissue containing the alpha-1B adrenergic receptor in rat spleen. | 19 | tissue-based format | Scientific Literature | |||
| 2. | ALA648011 | B | In vitro binding affinity towards alpha-1D adrenergic receptor of rat clone in radioligand binding assay | 52 | single protein format | Scientific Literature | |||
| 3. | ALA645471 | F | Efficacy relative to phenylephrine (PE) to constrict tissue containing the alpha-1A adrenergic receptor in rabbit urethra | Oryctolagus cuniculus | 29 | tissue-based format | Scientific Literature | ||
| 4. | ALA645473 | F | Functional agonism of the compounds to constrict tissue containing the alpha-1A adrenergic receptor in rabbit urethra | Oryctolagus cuniculus | 29 | tissue-based format | Scientific Literature | ||
| 5. | ALA648415 | B | In vitro binding affinity towards alpha-1A adrenergic receptor of rat submaxillary gland in radioligand binding assay | 46 | single protein format | Scientific Literature | |||
| 6. | ALA648102 | B | In vitro binding affinity towards alpha-1B adrenergic receptor of hamster clone in radioligand binding assay | Cricetulus griseus | 52 | single protein format | Scientific Literature | ||
| 7. | ALA663911 | F | Uroselectivity was determined by measuring effective dose required for 20 mmHg increase of mean arterial pressure (MAP) in vivo in dog; IA = Inactive | Canis lupus familiaris | 2 | organism-based format | Scientific Literature | ||
| 8. | ALA663913 | F | Uroselectivity was determined by measuring effective dose required for 5 mmHg increase of intraurethral pressure (IUP) in vivo in dog; IA = Inactive | Canis lupus familiaris | 2 | organism-based format | Scientific Literature | ||
| 9. | ALA845024 | B | Selectivity is ratio of pKi (binding affinity) of alpha-1B receptor to that of alpha-1A receptor. | 47 | protein format | Scientific Literature | |||
| 10. | ALA845025 | B | Selectivity is ratio of pKi (binding affinity) of Alpha-1D to that of alpha1A | 47 | protein format | Scientific Literature | |||
| 11. | ALA3057222 | B | Agonist activity at alpha1A adrenoreceptor in Oryctolagus cuniculus (rabbit) urethra relative to phenylephrine | Oryctolagus cuniculus | 17 | single protein format | Scientific Literature | ||
| 12. | ALA3056709 | B | Agonist activity at alpha1B adrenoreceptor in Rattus norvegicus (rat) spleen | Rattus norvegicus | 21 | single protein format | Scientific Literature | ||
| 13. | ALA3056710 | B | Binding affinity to Rattus norvegicus (rat) alpha1D adrenoreceptor by radioligand displacement assay | Rattus norvegicus | 30 | single protein format | Scientific Literature | ||
| 14. | ALA3056711 | B | Agonist activity at alpha1A adrenoreceptor in Oryctolagus cuniculus (rabbit) urethra | Oryctolagus cuniculus | 21 | single protein format | Scientific Literature | ||
| 15. | ALA3056712 | B | Binding affinity to alpha1A adrenoreceptor in Rattus norvegicus (rat) submaxillary gland by radioligand displacement assay | Rattus norvegicus | 30 | single protein format | Scientific Literature | ||
| 16. | ALA3056713 | B | Binding affinity to Cricetinae (hamster) alpha1B adrenoreceptor by radioligand displacement assay | Cricetinae | 30 | single protein format | Scientific Literature |
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