| # | Aladdin ID | Assay Type | Description | Organism | Compounds | Reference | BAO Format | Source | |
|---|---|---|---|---|---|---|---|---|---|
| 1. | ALA646233 | F | Functional agonism of the compounds to constrict tissue containing the alpha-1B adrenergic receptor in rat spleen | 10 | tissue-based format | Scientific Literature | |||
| 2. | ALA648011 | B | In vitro binding affinity towards alpha-1D adrenergic receptor of rat clone in radioligand binding assay | 52 | single protein format | Scientific Literature | |||
| 3. | ALA643232 | B | In vitro binding affinity towards alpha-2A adrenergic receptor of human clone in radioligand binding assay | 15 | single protein format | Scientific Literature | |||
| 4. | ALA643882 | F | Efficacy relative to phenylephrine (PE) to constrict tissue containing the alpha-2A adrenergic receptor in rat prostatic vas deferens | 11 | tissue-based format | Scientific Literature | |||
| 5. | ALA645786 | F | Functional agonism to constrict tissue containing alpha-2A adrenergic receptor in rat prostatic vas deferens | Rattus norvegicus | 10 | tissue-based format | Scientific Literature | ||
| 6. | ALA857772 | B | In vitro binding affinity towards alpha-2B adrenergic receptor of rat neonatal lung in radioligand binding assay | 15 | single protein format | Scientific Literature | |||
| 7. | ALA645471 | F | Efficacy relative to phenylephrine (PE) to constrict tissue containing the alpha-1A adrenergic receptor in rabbit urethra | Oryctolagus cuniculus | 29 | tissue-based format | Scientific Literature | ||
| 8. | ALA645473 | F | Functional agonism of the compounds to constrict tissue containing the alpha-1A adrenergic receptor in rabbit urethra | Oryctolagus cuniculus | 29 | tissue-based format | Scientific Literature | ||
| 9. | ALA648415 | B | In vitro binding affinity towards alpha-1A adrenergic receptor of rat submaxillary gland in radioligand binding assay | 46 | single protein format | Scientific Literature | |||
| 10. | ALA648102 | B | In vitro binding affinity towards alpha-1B adrenergic receptor of hamster clone in radioligand binding assay | Cricetulus griseus | 52 | single protein format | Scientific Literature | ||
| 11. | ALA647274 | F | Efficacy relative to phenylephrine (PE) constriction of rat spleen containing alpha-1B adrenergic receptor | Rattus norvegicus | 9 | tissue-based format | Scientific Literature | ||
| 12. | ALA663910 | F | Uroselectivity was determined by measuring effective dose required for 20 mmHg increase of mean arterial pressure (MAP) in vivo in dog | Canis lupus familiaris | 21 | organism-based format | Scientific Literature | ||
| 13. | ALA663912 | F | Uroselectivity was determined by measuring effective dose required for 5 mmHg increase of intraurethral pressure (IUP) in vivo in dog | Canis lupus familiaris | 21 | organism-based format | Scientific Literature | ||
| 14. | ALA849927 | F | Ratio of IUP ED delta5 to that of MAP ED delta20 | Canis lupus familiaris | 21 | organism-based format | Scientific Literature | ||
| 15. | ALA845021 | F | Selectivity is ratio of efficacy of alpha-2A to that of alpha1A adrenoceptor | 11 | assay format | Scientific Literature | |||
| 16. | ALA845022 | B | Relative affinities for alpha2B and alpha1A receptors | Rattus norvegicus | 15 | assay format | Scientific Literature | ||
| 17. | ALA845023 | B | Relative affinities for alpha-2a and alpha-1A receptors | 15 | assay format | Scientific Literature | |||
| 18. | ALA845024 | B | Selectivity is ratio of pKi (binding affinity) of alpha-1B receptor to that of alpha-1A receptor. | 47 | protein format | Scientific Literature | |||
| 19. | ALA845025 | B | Selectivity is ratio of pKi (binding affinity) of Alpha-1D to that of alpha1A | 47 | protein format | Scientific Literature | |||
| 20. | ALA3057220 | B | Agonist activity at alpha1B adrenoreceptor in Rattus norvegicus (rat) spleen relative to phenylephrine | Rattus norvegicus | 10 | single protein format | Scientific Literature |
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