# | Aladdin ID | Assay Type | Description | Organism | Compounds | Reference | BAO Format | Source | |
---|---|---|---|---|---|---|---|---|---|
1. | ALA3378283 | B | Inhibition of recombinant PDHK1 (unknown origin) expressed in Escherichia coli at 10 uM incubated for 1 hr by ELISA | Homo sapiens | 28 | ALA3352550 | assay format | Scientific Literature | |
2. | ALA3378284 | B | Inhibition of recombinant PDHK1 (unknown origin) expressed in Escherichia coli incubated for 1 hr by ELISA | Homo sapiens | 28 | ALA3352550 | assay format | Scientific Literature | |
3. | ALA3378285 | B | Inhibition of geldanamycin-BODIPY binding to full-length HSP90 (unknown origin) by fluorescence polarization based competition assay | Homo sapiens | 28 | ALA3352550 | protein format | Scientific Literature | |
4. | ALA3378286 | B | Inhibition of HSP90 in human NCI-H1299 cells assessed as reduction in AKT protein levels at 10 uM incubated for 12 hrs by immunoblotting method | Homo sapiens | 6 | ALA3352550 | cell-based format | Scientific Literature | |
5. | ALA3378287 | B | Inhibition of HSP90 in human NCI-H1299 cells assessed as reduction in HER2 protein levels at 10 uM incubated for 12 hrs by immunoblotting method | Homo sapiens | 6 | ALA3352550 | cell-based format | Scientific Literature | |
6. | ALA3378288 | B | Inhibition of HSP90 in human NCI-H1299 cells assessed as reduction in c-MET protein levels at 10 uM incubated for 12 hrs by immunoblotting method | Homo sapiens | 6 | ALA3352550 | cell-based format | Scientific Literature | |
7. | ALA3378289 | B | Inhibition of HSP90 in human NCI-H1299 cells assessed as increase in HSP70 protein levels at 10 uM incubated for 12 hrs by immunoblotting method | Homo sapiens | 6 | ALA3352550 | cell-based format | Scientific Literature | |
8. | ALA3378290 | A | Apparent permeability from apical to basolateral side in human Caco2 cells | Homo sapiens | 5 | ALA3352550 | cell-based format | Scientific Literature | |
9. | ALA3378291 | A | Apparent permeability from basolateral to apical side in human Caco2 cells | Homo sapiens | 5 | ALA3352550 | cell-based format | Scientific Literature | |
10. | ALA3378292 | A | Efflux ratio in human Caco2 cells | Homo sapiens | 5 | ALA3352550 | cell-based format | Scientific Literature | |
11. | ALA3378293 | B | Competitive Inhibition of recombinant PDHK1 (unknown origin) expressed in Escherichia coli incubated for 1 hr using varying ATP levels by by Lineweaver-Burk plot | Homo sapiens | 1 | ALA3352550 | assay format | Scientific Literature | |
12. | ALA3378294 | B | Inhibition of recombinant PDHK2 (unknown origin) expressed in Escherichia coli incubated for 1 hr by ELISA | Homo sapiens | 1 | ALA3352550 | assay format | Scientific Literature | |
13. | ALA3378295 | B | Inhibition of recombinant PDHK3 (unknown origin) expressed in Escherichia coli incubated for 1 hr by ELISA | Homo sapiens | 1 | ALA3352550 | assay format | Scientific Literature | |
14. | ALA3378296 | B | Inhibition of recombinant PDHK4 (unknown origin) expressed in Escherichia coli incubated for 1 hr by ELISA | Homo sapiens | 1 | ALA3352550 | assay format | Scientific Literature | |
15. | ALA3378297 | B | Inhibition of PDHK1 S293 phosphorylation in human NCI-H1299 cells incubated for 12 hrs by immunoblot | Homo sapiens | 1 | ALA3352550 | cell-based format | Scientific Literature | |
16. | ALA3378298 | B | Inhibition of PDHK1 S232 phosphorylation in human NCI-H1299 cells incubated for 12 hrs by immunoblot | Homo sapiens | 1 | ALA3352550 | cell-based format | Scientific Literature | |
17. | ALA3378851 | B | Inhibition of PDHK1 S293 phosphorylation in human NCI-H1299 cells incubated for 12 hrs by immunoblot relative to DCA | Homo sapiens | 1 | ALA3352550 | cell-based format | Scientific Literature | |
18. | ALA3378852 | B | Inhibition of PDHK1 S232 phosphorylation in human NCI-H1299 cells incubated for 12 hrs by immunoblot relative to DCA | Homo sapiens | 1 | ALA3352550 | cell-based format | Scientific Literature | |
19. | ALA3378853 | B | Inhibition of PDHK1 in human NCI-H1299 cells assessed as reduction in lactate production at 10 uM incubated for 12 hrs | Homo sapiens | 1 | ALA3352550 | cell-based format | Scientific Literature | |
20. | ALA3378855 | F | Reduction in extracellular acidification rate in human NCI-H1299 cells at 10 uM incubated for 12 hrs | Homo sapiens | 1 | ALA3352550 | cell-based format | Scientific Literature |