| # | Aladdin ID | Assay Type | Description | Organism | Compounds | Reference | BAO Format | Source | |
|---|---|---|---|---|---|---|---|---|---|
| 1. | ALA3378881 | B | Inhibition of human recombinant matriptase using Boc-Gln-Ala-Arg-AMC as substrate by microplate reader analysis | Homo sapiens | 15 | single protein format | Scientific Literature | ||
| 2. | ALA3371671 | B | Inhibition of human recombinant matriptase-2 using Boc-Gln-Ala-Arg-AMC as substrate by microplate reader analysis | Homo sapiens | 15 | single protein format | Scientific Literature | ||
| 3. | ALA3371672 | B | Selectivity ratio of Ki for human recombinant matriptase-2 to Ki for human recombinant matriptase | Homo sapiens | 15 | assay format | Scientific Literature | ||
| 4. | ALA3371673 | B | Selectivity ratio of Ki for human recombinant matriptase to Ki for human recombinant matriptase-2 | Homo sapiens | 3 | assay format | Scientific Literature | ||
| 5. | ALA4009362 | A | Stability in mouse plasma assessed as parent compound remaining after 24 hrs | Mus musculus | 4 | cell-free format | Scientific Literature | ||
| 6. | ALA4009363 | B | Inhibition of recombinant human C-terminal V5-His-tagged matriptase-2 expressed in Drosophila S2 cells using Boc-Gln-Ala-ArgAMC as substrate measured for 1200 mins by fluorescence assay | Homo sapiens | 29 | cell-based format | Scientific Literature | ||
| 7. | ALA4009364 | A | Inhibition of recombinant human matriptase (596 to 855 residues) expressed in Escherichia coli using Boc-Gln-Ala-ArgAMC as substrate measured for 1200 mins by fluorescence assay | Homo sapiens | 29 | assay format | Scientific Literature | ||
| 8. | ALA4009365 | B | Selectivity ratio of Ki for recombinant human matriptase (596 to 855 residues) expressed in Escherichia coli to Ki for recombinant human C-terminal V5-His-tagged matriptase-2 expressed in Drosophila S2 cells | Homo sapiens | 29 | cell-based format | Scientific Literature |
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