| # | Aladdin ID | Assay Type | Description | Organism | Compounds | Reference | BAO Format | Source | |
|---|---|---|---|---|---|---|---|---|---|
| 1. | ALA3388707 | B | Inhibition of human recombinant MMP13 using Cy3-PLGLK(Cy5Q)AR-NH2 as substrate after 40 mins by spectrofluorimetry | Homo sapiens | 37 | single protein format | Scientific Literature | ||
| 2. | ALA3388708 | B | Inhibition of human recombinant MMP1 using Cy3-PLGLK(Cy5Q)AR-NH2 as substrate after 40 mins by spectrofluorimetry | Homo sapiens | 3 | single protein format | Scientific Literature | ||
| 3. | ALA3388709 | B | Inhibition of human recombinant MMP2 using Cy3-PLGLK(Cy5Q)AR-NH2 as substrate after 40 mins by spectrofluorimetry | Homo sapiens | 3 | single protein format | Scientific Literature | ||
| 4. | ALA3388710 | B | Inhibition of human recombinant MMP3 using Cy3-PLGLK(Cy5Q)AR-NH2 as substrate after 40 mins by spectrofluorimetry | Homo sapiens | 3 | single protein format | Scientific Literature | ||
| 5. | ALA3388711 | B | Inhibition of human recombinant MMP7 using Cy3-PLGLK(Cy5Q)AR-NH2 as substrate after 40 mins by spectrofluorimetry | Homo sapiens | 3 | single protein format | Scientific Literature | ||
| 6. | ALA3388712 | B | Inhibition of human recombinant MMP8 using Cy3-PLGLK(Cy5Q)AR-NH2 as substrate after 40 mins by spectrofluorimetry | Homo sapiens | 3 | single protein format | Scientific Literature | ||
| 7. | ALA3388713 | B | Inhibition of human recombinant MMP9 using Cy3-PLGLK(Cy5Q)AR-NH2 as substrate after 40 mins by spectrofluorimetry | Homo sapiens | 3 | single protein format | Scientific Literature | ||
| 8. | ALA3389268 | B | Inhibition of human recombinant MMP10 using Cy3-PLGLK(Cy5Q)AR-NH2 as substrate after 40 mins by spectrofluorimetry | Homo sapiens | 3 | single protein format | Scientific Literature | ||
| 9. | ALA3389269 | B | Inhibition of human recombinant GST-tagged MMP14 using Cy3-PLGLK(Cy5Q)AR-NH2 as substrate after 40 mins by spectrofluorimetry | Homo sapiens | 3 | single protein format | Scientific Literature | ||
| 10. | ALA3389270 | B | Inhibition of human recombinant TACE using Cy3-PLAQAV(Cy5Q-L-2,3-diaminopropionic acid)-RSSSRNH2 as substrate after 40 mins by spectrofluorimetry | Homo sapiens | 3 | single protein format | Scientific Literature | ||
| 11. | ALA3389271 | A | Intrinsic clearance in iv dosed rat | Rattus norvegicus | 5 | organism-based format | Scientific Literature | ||
| 12. | ALA3389272 | A | Metabolic stability in rat liver microsomes | Rattus norvegicus | 5 | assay format | Scientific Literature | ||
| 13. | ALA3389313 | B | Selectivity ratio of IC50 for human recombinant MMP1 to IC50 for human recombinant MMP13 | Homo sapiens | 1 | assay format | Scientific Literature | ||
| 14. | ALA3389314 | B | Selectivity ratio of IC50 for human recombinant MMP2 to IC50 for human recombinant MMP13 | Homo sapiens | 1 | assay format | Scientific Literature | ||
| 15. | ALA3389315 | B | Selectivity ratio of IC50 for human recombinant MMP3 to IC50 for human recombinant MMP13 | Homo sapiens | 1 | assay format | Scientific Literature | ||
| 16. | ALA3389316 | B | Selectivity ratio of IC50 for human recombinant MMP7 to IC50 for human recombinant MMP13 | Homo sapiens | 1 | assay format | Scientific Literature | ||
| 17. | ALA3389317 | B | Selectivity ratio of IC50 for human recombinant MMP9 to IC50 for human recombinant MMP13 | Homo sapiens | 1 | assay format | Scientific Literature | ||
| 18. | ALA3389318 | B | Selectivity ratio of IC50 for human recombinant GAT-tagged MMP14 to IC50 for human recombinant MMP13 | Homo sapiens | 1 | assay format | Scientific Literature | ||
| 19. | ALA3389841 | A | Inhibition of cytochrome P450 (unknown origin) | Homo sapiens | 1 | assay format | Scientific Literature | ||
| 20. | ALA3389842 | B | Inhibition of human ERG | Homo sapiens | 1 | single protein format | Scientific Literature |
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