| # | Aladdin ID | Assay Type | Description | Organism | Compounds | Reference | BAO Format | Source | |
|---|---|---|---|---|---|---|---|---|---|
| 1. | ALA3384229 | F | Reduction in EED protein expression in human Toledo cells at 10 uM after 72 hrs by Western blot analysis | Homo sapiens | 1 | ALA3351265 | cell-based format | Scientific Literature | |
| 2. | ALA3384230 | F | Reduction in EZH2 protein expression in human Toledo cells at 10 uM after 72 hrs by Western blot analysis | Homo sapiens | 1 | ALA3351265 | cell-based format | Scientific Literature | |
| 3. | ALA3384231 | F | Reduction in SUZ12 protein expression in human Toledo cells at 10 uM after 72 hrs by Western blot analysis | Homo sapiens | 1 | ALA3351265 | cell-based format | Scientific Literature | |
| 4. | ALA3384232 | F | Reduction in EED protein expression in human DB cells at 10 uM after 72 hrs by Western blot analysis | Homo sapiens | 1 | ALA3351265 | cell-based format | Scientific Literature | |
| 5. | ALA3384233 | F | Reduction in EZH2 protein expression in human DB cells at 10 uM after 72 hrs by Western blot analysis | Homo sapiens | 1 | ALA3351265 | cell-based format | Scientific Literature | |
| 6. | ALA3384234 | F | Reduction in SUZ12 protein expression in human DB cells at 10 uM after 72 hrs by Western blot analysis | Homo sapiens | 1 | ALA3351265 | cell-based format | Scientific Literature | |
| 7. | ALA3421437 | B | Selectivity for human EZH2 over human GLP | Homo sapiens | 1 | ALA3414551 | assay format | Scientific Literature | |
| 8. | ALA3421438 | B | Selectivity for human EZH2 over human G9a | Homo sapiens | 1 | ALA3414551 | assay format | Scientific Literature | |
| 9. | ALA3421439 | B | Competitive inhibition of human EZH2 using SAM and histone H3 (16 to 30) as substrate preincubated for 30 mins followed by substrate addition measured after 90 mins by Michaelis-Menten plot analysis | Homo sapiens | 1 | ALA3414551 | single protein format | Scientific Literature | |
| 10. | ALA3421440 | B | Inhibition of human EZH2 using SAM and histone H3 (16 to 30) as substrate preincubated for 30 mins followed by substrate addition measured after 90 mins by flash plate assay | Homo sapiens | 2 | ALA3414551 | single protein format | Scientific Literature | |
| 11. | ALA3421449 | B | Selectivity for human EZH2 over human SETD7 | Homo sapiens | 1 | ALA3414551 | assay format | Scientific Literature | |
| 12. | ALA3421450 | B | Selectivity for human EZH2 over human SMYD2 | Homo sapiens | 1 | ALA3414551 | assay format | Scientific Literature | |
| 13. | ALA3421451 | B | Selectivity for human EZH2 over human SMYD3 | Homo sapiens | 1 | ALA3414551 | assay format | Scientific Literature | |
| 14. | ALA3421452 | B | Selectivity for human EZH2 over human WHSC1L1 | Homo sapiens | 1 | ALA3414551 | assay format | Scientific Literature | |
| 15. | ALA3421453 | B | Selectivity for human EZH2 over human MMSET | Homo sapiens | 1 | ALA3414551 | assay format | Scientific Literature | |
| 16. | ALA3421454 | B | Selectivity for human EZH2 over human PRMT1 | Homo sapiens | 1 | ALA3414551 | assay format | Scientific Literature | |
| 17. | ALA3421455 | B | Selectivity for human EZH2 over human PRMT3 | Homo sapiens | 1 | ALA3414551 | assay format | Scientific Literature | |
| 18. | ALA3421456 | B | Selectivity for human EZH2 over human PRMT4 | Homo sapiens | 1 | ALA3414551 | assay format | Scientific Literature | |
| 19. | ALA3421457 | B | Selectivity for human EZH2 over human PRMT5 | Homo sapiens | 1 | ALA3414551 | assay format | Scientific Literature | |
| 20. | ALA3421458 | B | Selectivity for human EZH2 over human PRMT6 | Homo sapiens | 1 | ALA3414551 | assay format | Scientific Literature |
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