# | Aladdin ID | Assay Type | Description | Organism | Compounds | Reference | BAO Format | Source | |
---|---|---|---|---|---|---|---|---|---|
1. | ALA3387185 | Binding | Displacement of [3H]NPVF from human NPFF1 receptor expressed in CHO cells after 1 hr by liquid scintillation counting analysis | Homo sapiens | 25 | ALA3351542 | cell-based format | Scientific Literature | |
2. | ALA3387186 | Binding | Displacement of [3H]EYF from human NPFF2 receptor expressed in CHO cells after 1 hr by liquid scintillation counting analysis | Homo sapiens | 29 | ALA3351542 | cell-based format | Scientific Literature | |
3. | ALA3387188 | Binding | Selectivity ratio of Ki for human NPFF1 receptor to Ki for human NPFF2 receptor | Homo sapiens | 8 | ALA3351542 | assay format | Scientific Literature | |
4. | ALA3387189 | Binding | Displacement of [3H]DAMGO from human MOR expressed in HEK293 cells after 60 mins by scintillation counting analysis | Homo sapiens | 8 | ALA3351542 | cell-based format | Scientific Literature | |
5. | ALA3387190 | Binding | Displacement of [3H]DPDPE from human DOR expressed in HEK293 cells after 60 mins by scintillation counting analysis | Homo sapiens | 8 | ALA3351542 | cell-based format | Scientific Literature | |
6. | ALA3387191 | Binding | Displacement of [3H]U-69593 from human KOR expressed in HEK293 cells after 60 mins by scintillation counting analysis | Homo sapiens | 8 | ALA3351542 | cell-based format | Scientific Literature | |
7. | ALA3387755 | Functional | Antagonist activity at human NPFF1 receptor expressed in CHO cells assessed as reversal of NPVF-induced inhibition of intracellular cAMP accumulation after 10 mins by liquid scintillation counting analysis relative to control | Homo sapiens | 3 | ALA3351542 | cell-based format | Scientific Literature | |
8. | ALA3387759 | Functional | Antagonist activity at human NPFF2 receptor expressed in CHO cells assessed as reversal of 1DMe-induced inhibition of intracellular cAMP accumulation after 10 mins by liquid scintillation counting analysis relative to control | Homo sapiens | 1 | ALA3351542 | cell-based format | Scientific Literature | |
9. | ALA3387760 | Binding | Partial antagonist activity at human NPFF1 receptor expressed in CHO cells assessed NPVF EC50 at 10 uM after 10 mins by liquid scintillation counting analysis to NPVF EC50 alone | Homo sapiens | 1 | ALA3351542 | cell-based format | Scientific Literature | |
10. | ALA3387761 | Binding | Partial antagonist activity at human NPFF2 receptor expressed in CHO cells assessed 1DMe EC50 at 10 uM after 10 mins by liquid scintillation counting analysis to 1DMe EC50 alone | Homo sapiens | 1 | ALA3351542 | cell-based format | Scientific Literature | |
11. | ALA3387765 | Binding | Selectivity ratio of Ki for human MOR to Ki for human NPFF2 receptor | Homo sapiens | 2 | ALA3351542 | assay format | Scientific Literature | |
12. | ALA3387766 | Binding | Selectivity ratio of Ki for human KOR to Ki for human NPFF2 receptor | Homo sapiens | 2 | ALA3351542 | assay format | Scientific Literature |