| # | Aladdin ID | Assay Type | Description | Organism | Compounds | Reference | BAO Format | Source | |
|---|---|---|---|---|---|---|---|---|---|
| 1. | ALA3396419 | B | Inhibition of full length recombinant Pim-1 (unknown origin) assessed as phosphorylation of biotinylated-BAD peptide at Serine 112 residue | Homo sapiens | 31 | ALA3392976 | single protein format | Scientific Literature | |
| 2. | ALA3396420 | B | Inhibition of full length recombinant Pim-2 (unknown origin) assessed as phosphorylation of biotinylated-BAD peptide at Serine 112 residue | Homo sapiens | 31 | ALA3392976 | single protein format | Scientific Literature | |
| 3. | ALA3396421 | B | Inhibition of full length recombinant Pim-3 (unknown origin) assessed as phosphorylation of biotinylated-BAD peptide at Serine 112 residue | Homo sapiens | 18 | ALA3392976 | single protein format | Scientific Literature | |
| 4. | ALA3396422 | B | Inhibition of pan Pim in human KMS-12-BM cells assessed as phosphorylation of biotinylated-BAD peptide | Homo sapiens | 14 | ALA3392976 | cell-based format | Scientific Literature | |
| 5. | ALA3396423 | A | Intrinsic clearance in rat liver microsomes assessed as compound remaining at 1 uM after 30 mins | Rattus norvegicus | 7 | ALA3392976 | assay format | Scientific Literature | |
| 6. | ALA3396424 | A | Clearance in Sprague-Dawley rat at 2 mg/kg, iv | Rattus norvegicus | 7 | ALA3392976 | organism-based format | Scientific Literature | |
| 7. | ALA3396425 | A | Volume of distribution at steady state in Sprague-Dawley rat at 2 mg/kg, iv | Rattus norvegicus | 7 | ALA3392976 | organism-based format | Scientific Literature | |
| 8. | ALA3396426 | A | Half life in Sprague-Dawley rat at 2 mg/kg, iv | Rattus norvegicus | 7 | ALA3392976 | organism-based format | Scientific Literature | |
| 9. | ALA3396427 | A | AUC in Sprague-Dawley rat at 5 mg/kg, po | Rattus norvegicus | 7 | ALA3392976 | organism-based format | Scientific Literature | |
| 10. | ALA3396428 | A | Oral bioavailability in Sprague-Dawley rat at 5 mg/kg | Rattus norvegicus | 7 | ALA3392976 | organism-based format | Scientific Literature | |
| 11. | ALA3396429 | B | Inhibition of human ERG | Homo sapiens | 7 | ALA3392976 | single protein format | Scientific Literature | |
| 12. | ALA3396430 | B | Competitive binding affinity at CAMK4 (unknown origin) at 1 uM relative to control | Homo sapiens | 1 | ALA3392976 | single protein format | Scientific Literature | |
| 13. | ALA3396431 | B | Competitive binding affinity at CLK2 (unknown origin) at 1 uM relative to control | Homo sapiens | 1 | ALA3392976 | single protein format | Scientific Literature | |
| 14. | ALA3396432 | B | Competitive binding affinity at CLK4 (unknown origin) at 1 uM relative to control | Homo sapiens | 1 | ALA3392976 | single protein format | Scientific Literature | |
| 15. | ALA3396433 | B | Competitive binding affinity at DMPK (unknown origin) at 1 uM relative to control | Homo sapiens | 1 | ALA3392976 | single protein format | Scientific Literature | |
| 16. | ALA3396434 | B | Competitive binding affinity at DYRK1A (unknown origin) at 1 uM relative to control | Homo sapiens | 1 | ALA3392976 | single protein format | Scientific Literature | |
| 17. | ALA3396435 | B | Competitive binding affinity at DYRK1B (unknown origin) at 1 uM relative to control | Homo sapiens | 1 | ALA3392976 | single protein format | Scientific Literature | |
| 18. | ALA3396436 | B | Competitive binding affinity at JAK2 (unknown origin) at 1 uM relative to control | Homo sapiens | 1 | ALA3392976 | single protein format | Scientific Literature | |
| 19. | ALA3396437 | B | Competitive binding affinity at MEK5 (unknown origin) at 1 uM relative to control | Homo sapiens | 1 | ALA3392976 | single protein format | Scientific Literature | |
| 20. | ALA3396438 | B | Competitive binding affinity at PIM1 (unknown origin) at 1 uM relative to control | Homo sapiens | 1 | ALA3392976 | single protein format | Scientific Literature |
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