| # | Aladdin ID | Assay Type | Description | Organism | Compounds | Reference | BAO Format | Source | |
|---|---|---|---|---|---|---|---|---|---|
| 1. | ALA3398933 | B | Inhibition of N-terminally FLAG-tagged wild type EZH2 in EZH2/SUZ12/EED/RbAp48 complex (unknown origin) expressed in baculovirus infected in SF9 cells assessed as inhibition of methylation of nucleosomes at H3K27 by scintillation counting in presence of [3H]SAM | Homo sapiens | 17 | cell-based format | Scientific Literature | ||
| 2. | ALA3399055 | B | Inhibition of N-terminally FLAG-tagged EZH2 Y641N mutant in EZH2/SUZ12/EED/RbAp48 complex (unknown origin) expressed in baculovirus infected in SF9 cells assessed as inhibition of methylation of nucleosomes at H3K27 by scintillation counting in presence of [3H]SAM | Homo sapiens | 12 | cell-based format | Scientific Literature | ||
| 3. | ALA3399056 | B | Inhibition of EZH2 (unknown origin) at 100 uM by cell-based assay | Homo sapiens | 2 | cell-based format | Scientific Literature | ||
| 4. | ALA3399057 | A | Permeability across MDCK2 cells | Canis lupus familiaris | 1 | cell-based format | Scientific Literature | ||
| 5. | ALA3399058 | B | Inhibition of EZH1 (unknown origin) by HMT assay | Homo sapiens | 2 | single protein format | Scientific Literature | ||
| 6. | ALA3399059 | B | Ratio of S-adenosyl-L-homocysteine IC50 to compound IC50 for N-terminally FLAG-tagged wild type EZH2 in EZH2/SUZ12/EED/RbAp48 complex (unknown origin) expressed in baculovirus infected in SF9 cells assessed as inhibition of methylation of nucleosomes at H3K27 at 20 uM by scintillation counting in presence of [3H]SAM | Homo sapiens | 1 | cell-based format | Scientific Literature | ||
| 7. | ALA3399060 | B | Inhibition of G9a (unknown origin) by HMT assay | Homo sapiens | 2 | single protein format | Scientific Literature | ||
| 8. | ALA3399061 | B | Inhibition of EHMT1 (unknown origin) by HMT assay | Homo sapiens | 2 | single protein format | Scientific Literature | ||
| 9. | ALA3399062 | B | Inhibition of MLL (unknown origin) by HMT assay | Homo sapiens | 2 | single protein format | Scientific Literature | ||
| 10. | ALA3399063 | B | Inhibition of SETD7 (unknown origin) by HMT assay | Homo sapiens | 2 | single protein format | Scientific Literature | ||
| 11. | ALA3399136 | B | Inhibition of SETDB1 (unknown origin) by HMT assay | Homo sapiens | 2 | single protein format | Scientific Literature | ||
| 12. | ALA3399137 | B | Inhibition of SUV39H1 (unknown origin) by HMT assay | Homo sapiens | 2 | single protein format | Scientific Literature | ||
| 13. | ALA3399138 | B | Inhibition of SUV39H2 (unknown origin) by HMT assay | Homo sapiens | 2 | single protein format | Scientific Literature | ||
| 14. | ALA3399139 | B | Inhibition of SUV420H2 (unknown origin) by HMT assay | Homo sapiens | 2 | single protein format | Scientific Literature | ||
| 15. | ALA3399140 | B | Inhibition of SMYD2 (unknown origin) by HMT assay | Homo sapiens | 2 | single protein format | Scientific Literature | ||
| 16. | ALA3399141 | B | Inhibition of G9a (unknown origin) at 10 uM by HMT assay | Homo sapiens | 1 | single protein format | Scientific Literature | ||
| 17. | ALA3399142 | B | Inhibition of EHMT1 (unknown origin) at 10 uM by HMT assay | Homo sapiens | 1 | single protein format | Scientific Literature | ||
| 18. | ALA3399143 | B | Inhibition of SETD7 (unknown origin) at 10 uM by HMT assay | Homo sapiens | 1 | single protein format | Scientific Literature | ||
| 19. | ALA3399144 | B | Inhibition of SETDB1 (unknown origin) at 10 uM by HMT assay | Homo sapiens | 1 | single protein format | Scientific Literature | ||
| 20. | ALA3399145 | B | Inhibition of SUV39H2 (unknown origin) at 10 uM by HMT assay | Homo sapiens | 1 | single protein format | Scientific Literature |
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