| # | Aladdin ID | Assay Type | Description | Organism | Compounds | Reference | BAO Format | Source | |
|---|---|---|---|---|---|---|---|---|---|
| 1. | ALA3398862 | A | Half life in sc dosed rat | Rattus norvegicus | 1 | ALA3397017 | organism-based format | Scientific Literature | |
| 2. | ALA3398863 | F | Prevention of right ventricular weight increase in rat model of monocrotaline-induced pulmonary arterial hypertension administered subcutaneously twice daily for 21 days | Rattus norvegicus | 1 | ALA3397017 | organism-based format | Scientific Literature | |
| 3. | ALA3398864 | F | Prevention of right ventricular weight increase in rat model of monocrotaline-induced pulmonary arterial hypertension at 30 mg/kg, sc administered twice daily for 21 days relative to sham animal (Rvb = 19 no unit) | Rattus norvegicus | 2 | ALA3397017 | organism-based format | Scientific Literature | |
| 4. | ALA3398865 | F | Prevention of right ventricular weight increase in rat model of monocrotaline-induced pulmonary arterial hypertension at 10 mg/kg, sc administered twice daily for 21 days relative to sham animal (Rvb = 19 no unit) | Rattus norvegicus | 2 | ALA3397017 | organism-based format | Scientific Literature | |
| 5. | ALA3398866 | F | Prevention of right ventricular weight increase in rat model of monocrotaline-induced pulmonary arterial hypertension at 1 mg/kg, sc administered twice daily for 21 days relative to sham animal (Rvb = 19 no unit) | Rattus norvegicus | 1 | ALA3397017 | organism-based format | Scientific Literature | |
| 6. | ALA3398867 | F | Improvement in right ventricular systolic pressure in rat model of monocrotaline-induced pulmonary arterial hypertension at 10 mg/kg, sc administered twice daily for 21 days | Rattus norvegicus | 1 | ALA3397017 | organism-based format | Scientific Literature | |
| 7. | ALA3398868 | F | Agonist activity at human recombinant DP1 receptor by cAMP assay | Homo sapiens | 2 | ALA3397017 | single protein format | Scientific Literature | |
| 8. | ALA3398869 | B | Selectivity index, ratio of EC50 for human recombinant DP1 receptor to EC50 for human recombinant IP receptor | Homo sapiens | 1 | ALA3397017 | assay format | Scientific Literature | |
| 9. | ALA3399046 | F | Agonist activity at human recombinant IP receptor expressed in CHO-K1 cells incubated for 1 hr by HTRF cAMP assay | Homo sapiens | 32 | ALA3397017 | cell-based format | Scientific Literature | |
| 10. | ALA3399047 | F | Intrinsic activity at human recombinant IP receptor expressed in CHO-K1 cells incubated for 1 hr by HTRF cAMP assay relative to 1 uM iloprost | Homo sapiens | 32 | ALA3397017 | cell-based format | Scientific Literature | |
| 11. | ALA3399048 | F | Agonist activity at rat recombinant IP receptor expressed in CHO-K1 cells incubated for 1 hr by HTRF cAMP assay | Rattus norvegicus | 32 | ALA3397017 | cell-based format | Scientific Literature | |
| 12. | ALA3399049 | F | Intrinsic activity at rat recombinant IP receptor expressed in CHO-K1 cells incubated for 1 hr by HTRF cAMP assay relative to 1 uM iloprost | Rattus norvegicus | 32 | ALA3397017 | cell-based format | Scientific Literature | |
| 13. | ALA3399050 | B | Agonist activity at human recombinant DP1 receptor expressed in melanophores assessed as induction of pigment redistribution incubated for 90 mins | Homo sapiens | 32 | ALA3397017 | assay format | Scientific Literature | |
| 14. | ALA3399051 | B | Agonist activity at human IP receptor in human platelets assessed as inhibition of ADP-induced platelet aggregation | Homo sapiens | 16 | ALA3397017 | assay format | Scientific Literature | |
| 15. | ALA3399052 | A | Stability in rat liver microsomes | Rattus norvegicus | 13 | ALA3397017 | assay format | Scientific Literature | |
| 16. | ALA3399053 | A | Stability in human liver microsomes | Homo sapiens | 13 | ALA3397017 | assay format | Scientific Literature |
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