# | Aladdin ID | Assay Type | Description | Organism | Compounds | Reference | BAO Format | Source | |
---|---|---|---|---|---|---|---|---|---|
1. | ALA3413938 | B | Inhibition of human KLK7 using Suc-Leu-Leu-Val-Tyr-AMC as substrate after 15 mins by fluorescence assay | Homo sapiens | 11 | ALA3407351 | single protein format | Scientific Literature | |
2. | ALA3413940 | B | Competitive inhibition of human KLK7 using Suc-Leu-Leu-Val-Tyr-AMC as substrate by Lineweaver-Burk plot analysis | Homo sapiens | 2 | ALA3407351 | single protein format | Scientific Literature | |
3. | ALA3413941 | B | Inhibition of human KLK5 using Boc-Val-Pro-Arg-AMC as substrate at 50 uM after 15 mins by fluorescence assay | Homo sapiens | 2 | ALA3407351 | single protein format | Scientific Literature | |
4. | ALA3413942 | B | Inhibition of human KLK8 using Boc-Val-Pro-Arg-AMC as substrate at 50 uM after 15 mins by fluorescence assay | Homo sapiens | 2 | ALA3407351 | single protein format | Scientific Literature | |
5. | ALA3413943 | B | Inhibition of human KLK14 using Boc-Val-Pro-Arg-AMC as substrate at 50 uM after 15 mins by fluorescence assay | Homo sapiens | 2 | ALA3407351 | single protein format | Scientific Literature | |
6. | ALA3413944 | B | Reversible inhibition of human KLK7 using Suc-Leu-Leu-Val-Tyr-AMC as substrate at 50 uM preincubated for 15 mins followed by 40 fold dilution by fluorescence assay | Homo sapiens | 1 | ALA3407351 | single protein format | Scientific Literature | |
7. | ALA3413945 | F | Cytotoxicity against human HeLa cells assessed as cell death after 48 to 72 hrs by XTT assay | Homo sapiens | 4 | ALA3407351 | cell-based format | Scientific Literature | |
8. | ALA3413946 | F | Cytotoxicity against human PC3 cells assessed as cell death after 48 to 72 hrs by XTT assay | Homo sapiens | 4 | ALA3407351 | cell-based format | Scientific Literature | |
9. | ALA3414068 | F | Cytotoxicity against human SW620 cells assessed as cell death after 48 to 72 hrs by XTT assay | Homo sapiens | 4 | ALA3407351 | cell-based format | Scientific Literature |