| # | Aladdin ID | Assay Type | Description | Organism | Compounds | Reference | BAO Format | Source | |
|---|---|---|---|---|---|---|---|---|---|
| 1. | ALA3418470 | B | Inhibition of EZH2 (unknown origin) using biotinylated-histone H3 (1 to 24) as substrate after 1 hr by scintillation proximity assay in presence of [3H]-SAM | Homo sapiens | 3 | single protein format | Scientific Literature | ||
| 2. | ALA3418471 | B | Competitive inhibition of EZH2 (unknown origin) using biotinylated-histone H3 (1 to 24) as substrate by Lineweaver-Burk plot analysis in presence of SAM | Homo sapiens | 1 | single protein format | Scientific Literature | ||
| 3. | ALA3418472 | B | Selectivity for EZH2 (unknown origin) over G9a (unknown origin) | Homo sapiens | 1 | assay format | Scientific Literature | ||
| 4. | ALA3418473 | B | Selectivity for EZH2 (unknown origin) over GLP (unknown origin) | Homo sapiens | 1 | assay format | Scientific Literature | ||
| 5. | ALA3418474 | B | Selectivity for EZH2 (unknown origin) over SUV39H2 (unknown origin) | Homo sapiens | 1 | assay format | Scientific Literature | ||
| 6. | ALA3418475 | B | Selectivity for EZH2 (unknown origin) over SUV420H1 (unknown origin) | Homo sapiens | 1 | assay format | Scientific Literature | ||
| 7. | ALA3418476 | B | Selectivity for EZH2 (unknown origin) over SUV420H2 (unknown origin) | Homo sapiens | 1 | assay format | Scientific Literature | ||
| 8. | ALA3418477 | B | Selectivity for EZH2 (unknown origin) over MLL1 (unknown origin) | Homo sapiens | 1 | assay format | Scientific Literature | ||
| 9. | ALA3418478 | B | Selectivity for EZH2 (unknown origin) over SETDB1 (unknown origin) | Homo sapiens | 1 | assay format | Scientific Literature | ||
| 10. | ALA3418479 | B | Selectivity for EZH2 (unknown origin) over SETD7 (unknown origin) | Homo sapiens | 1 | assay format | Scientific Literature | ||
| 11. | ALA3418480 | B | Selectivity for EZH2 (unknown origin) over SETD8 (unknown origin) | Homo sapiens | 1 | assay format | Scientific Literature | ||
| 12. | ALA3418481 | B | Selectivity for EZH2 (unknown origin) over SMYD2 (unknown origin) | Homo sapiens | 1 | assay format | Scientific Literature | ||
| 13. | ALA3418482 | B | Selectivity for EZH2 (unknown origin) over PRMT1 (unknown origin) | Homo sapiens | 1 | assay format | Scientific Literature | ||
| 14. | ALA3418483 | B | Selectivity for EZH2 (unknown origin) over PRMT3 (unknown origin) | Homo sapiens | 1 | assay format | Scientific Literature | ||
| 15. | ALA3418484 | B | Selectivity for EZH2 (unknown origin) over PRMT5 (unknown origin) | Homo sapiens | 1 | assay format | Scientific Literature | ||
| 16. | ALA3418485 | B | Selectivity for EZH2 (unknown origin) over DOT1L (unknown origin) | Homo sapiens | 1 | assay format | Scientific Literature | ||
| 17. | ALA3418487 | B | Selectivity for EZH2 (unknown origin) over DNMT1 (unknown origin) | Homo sapiens | 1 | assay format | Scientific Literature | ||
| 18. | ALA3418488 | B | Selectivity ratio of IC50 for EZH1 (unknown origin) to IC50 for EZH2 (unknown origin) | Homo sapiens | 1 | assay format | Scientific Literature | ||
| 19. | ALA3418489 | B | Inhibition of EZH2 in human MCF10A cells assessed as reduction of H3K27me3 level after 72 hrs by Western blot analysis | Homo sapiens | 1 | cell-based format | Scientific Literature | ||
| 20. | ALA3418668 | A | Cytotoxicity against human MCF10A cells assessed as cell viability by Alamar Blue assay | Homo sapiens | 1 | cell-based format | Scientific Literature |
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