| # | Aladdin ID | Assay Type | Description | Organism | Compounds | Reference | BAO Format | Source | |
|---|---|---|---|---|---|---|---|---|---|
| 1. | ALA3419341 | B | Inhibition of human NaV1.8 at -140 mV holding potential by whole-cell patch clamp assay | Homo sapiens | 1 | assay format | Scientific Literature | ||
| 2. | ALA3419342 | B | Inhibition of human NaV1.7 at -140 mV holding potential by whole-cell patch clamp assay | Homo sapiens | 70 | assay format | Scientific Literature | ||
| 3. | ALA3419343 | B | Inhibition of human NaV1.5 at -140 mV holding potential by whole-cell patch clamp assay | Homo sapiens | 70 | assay format | Scientific Literature | ||
| 4. | ALA3419344 | B | Inhibition of human NaV1.4 at -140 mV holding potential by whole-cell patch clamp assay | Homo sapiens | 70 | assay format | Scientific Literature | ||
| 5. | ALA3419345 | B | Inhibition of human NaV1.3 at -140 mV holding potential by whole-cell patch clamp assay | Homo sapiens | 1 | assay format | Scientific Literature | ||
| 6. | ALA3419346 | B | Inhibition of NaV1.7 in C57BL/6 mouse DRG neurons at -140 mV holding potential by whole-cell patch clamp assay | Mus musculus | 2 | assay format | Scientific Literature | ||
| 7. | ALA3419347 | B | Inhibition of NaV1.7 in C57BL/6 mouse DRG neurons held at voltage yielding 20% inactivation and depolarized to -10 mV for 40 ms every 10 s by whole-cell patch clamp assay | Mus musculus | 1 | assay format | Scientific Literature | ||
| 8. | ALA3419348 | B | Selectivity index, ratio of IC50 for human NaV1.5 to IC50 for human NaV1.7 | Homo sapiens | 10 | assay format | Scientific Literature | ||
| 9. | ALA3419349 | B | Selectivity index, ratio of IC50 for human NaV1.4 to IC50 for human NaV1.7 | Homo sapiens | 10 | assay format | Scientific Literature | ||
| 10. | ALA4321987 | B | Inhibition of human Nav1.7 expressed in HEK293 cells by electrophysiology assay | Homo sapiens | 15 | cell-based format | Scientific Literature | ||
| 11. | ALA4321994 | B | Inhibition of human Nav1.4 expressed in HEK293 cells by electrophysiology assay | Homo sapiens | 11 | cell-based format | Scientific Literature | ||
| 12. | ALA4321995 | B | Inhibition of human Nav1.5 expressed in HEK293 cells by electrophysiology assay | Homo sapiens | 14 | cell-based format | Scientific Literature | ||
| 13. | ALA4322001 | B | Selectivity index, ratio of IC50 for inhibition of human Nav1.4 expressed in HEK293 cells by electrophysiology assay to IC50 for inhibition of human Nav1.7 expressed in HEK293 cells by electrophysiology assay | Homo sapiens | 11 | cell-based format | Scientific Literature | ||
| 14. | ALA4322002 | B | Selectivity index, ratio of IC50 for inhibition of human Nav1.5 expressed in HEK293 cells by electrophysiology assay to IC50 for inhibition of human Nav1.7 expressed in HEK293 cells by electrophysiology assay | Homo sapiens | 14 | cell-based format | Scientific Literature |
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