| # | Aladdin ID | Assay Type | Description | Organism | Compounds | Reference | BAO Format | Source | |
|---|---|---|---|---|---|---|---|---|---|
| 1. | ALA3419342 | B | Inhibition of human NaV1.7 at -140 mV holding potential by whole-cell patch clamp assay | Homo sapiens | 70 | assay format | Scientific Literature | ||
| 2. | ALA3419343 | B | Inhibition of human NaV1.5 at -140 mV holding potential by whole-cell patch clamp assay | Homo sapiens | 70 | assay format | Scientific Literature | ||
| 3. | ALA3419344 | B | Inhibition of human NaV1.4 at -140 mV holding potential by whole-cell patch clamp assay | Homo sapiens | 70 | assay format | Scientific Literature | ||
| 4. | ALA3419346 | B | Inhibition of NaV1.7 in C57BL/6 mouse DRG neurons at -140 mV holding potential by whole-cell patch clamp assay | Mus musculus | 2 | assay format | Scientific Literature | ||
| 5. | ALA3419348 | B | Selectivity index, ratio of IC50 for human NaV1.5 to IC50 for human NaV1.7 | Homo sapiens | 10 | assay format | Scientific Literature | ||
| 6. | ALA3419349 | B | Selectivity index, ratio of IC50 for human NaV1.4 to IC50 for human NaV1.7 | Homo sapiens | 10 | assay format | Scientific Literature | ||
| 7. | ALA3419350 | B | Inhibition of human NaV1.7 by patchXpress 700A electrophysiology method | Homo sapiens | 1 | single protein format | Scientific Literature | ||
| 8. | ALA3419351 | B | Inhibition of human NaV1.4 by patchXpress 700A electrophysiology method | Homo sapiens | 1 | single protein format | Scientific Literature | ||
| 9. | ALA3419352 | B | Inhibition of human NaV1.7 assessed as reduction in peak inward current at -10 mV by manual whole cell patch clamp electrophysiology method | Homo sapiens | 1 | assay format | Scientific Literature | ||
| 10. | ALA3419510 | A | Stability in human plasma assessed as intact compound remaining at 37 degC after 24 hrs by LC-MS method | Homo sapiens | 1 | cell-free format | Scientific Literature | ||
| 11. | ALA3419511 | A | Stability in mouse plasma assessed as intact compound remaining at 37 degC after 24 hrs by LC-MS method | Mus musculus | 1 | cell-free format | Scientific Literature | ||
| 12. | ALA3803506 | B | Inhibition of human Nav1.7 expressed in HEK293 cells assessed as inward peak current by ion-works quattro patch clamp electrophysiology method | Homo sapiens | 160 | cell-based format | Scientific Literature | ||
| 13. | ALA3803507 | B | Inhibition of human Nav1.5 expressed in HEK293 cells assessed as inward peak current by ion-works quattro patch clamp electrophysiology method | Homo sapiens | 160 | cell-based format | Scientific Literature | ||
| 14. | ALA3803508 | B | Inhibition of human Nav1.4 expressed in HEK293 cells assessed as inward peak current by ion-works quattro patch clamp electrophysiology method | Homo sapiens | 160 | cell-based format | Scientific Literature |
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