| # | Aladdin ID | Assay Type | Description | Organism | Compounds | Reference | BAO Format | Source | |
|---|---|---|---|---|---|---|---|---|---|
| 1. | ALA3421047 | B | Binding affinity to human histamine H3 receptor | Homo sapiens | 10 | single protein format | Scientific Literature | ||
| 2. | ALA3421048 | B | Binding affinity to rat histamine H3 receptor | Rattus norvegicus | 10 | single protein format | Scientific Literature | ||
| 3. | ALA3421049 | A | Half life in mouse liver microsomes | Mus musculus | 4 | assay format | Scientific Literature | ||
| 4. | ALA3421050 | A | Half life in rat liver microsomes | Rattus norvegicus | 4 | assay format | Scientific Literature | ||
| 5. | ALA3421052 | A | Half life in monkey liver microsomes | Macaca mulatta | 4 | assay format | Scientific Literature | ||
| 6. | ALA3421053 | A | Half life in human liver microsomes | Homo sapiens | 4 | assay format | Scientific Literature | ||
| 7. | ALA3421054 | A | Inhibition of CYP1A2 (unknown origin) | Homo sapiens | 4 | single protein format | Scientific Literature | ||
| 8. | ALA3421055 | A | Inhibition of CYP2C9 (unknown origin) | Homo sapiens | 4 | single protein format | Scientific Literature | ||
| 9. | ALA3421056 | A | Inhibition of CYP2C19 (unknown origin) | Homo sapiens | 4 | single protein format | Scientific Literature | ||
| 10. | ALA3421057 | A | Inhibition of CYP2D6 (unknown origin) | Homo sapiens | 4 | single protein format | Scientific Literature | ||
| 11. | ALA3421058 | A | Inhibition of CYP3A4 (unknown origin) | Homo sapiens | 4 | single protein format | Scientific Literature | ||
| 12. | ALA3421063 | F | Antagonist activity at human H3R expressed in CHO cells assessed as inhibition of RAMH-induced [35S]GTPgammaS binding relative to control | Homo sapiens | 2 | cell-based format | Scientific Literature | ||
| 13. | ALA3421064 | B | Inhibition of human H1R | Homo sapiens | 2 | single protein format | Scientific Literature | ||
| 14. | ALA3421065 | B | Inhibition of human H2R | Homo sapiens | 2 | single protein format | Scientific Literature | ||
| 15. | ALA3421066 | B | Inhibition of human H4R | Homo sapiens | 2 | single protein format | Scientific Literature | ||
| 16. | ALA3421067 | B | Inhibition of DAT (unknown origin) | Homo sapiens | 2 | single protein format | Scientific Literature | ||
| 17. | ALA3421068 | B | Inhibition of alpha-2C adrenergic receptor (unknown origin) | Homo sapiens | 2 | single protein format | Scientific Literature | ||
| 18. | ALA3421069 | B | Selectivity ratio of Ki for DAT (unknown origin) to Ki for human histamine H3 receptor | Homo sapiens | 2 | assay format | Scientific Literature | ||
| 19. | ALA3421070 | B | Selectivity ratio of Ki for alpha-2C adrenergic receptor (unknown origin) to Ki for human histamine H3 receptor | Homo sapiens | 2 | assay format | Scientific Literature | ||
| 20. | ALA3421071 | P | Aqueous solubility of the compound at pH 7.4 | 2 | small-molecule physicochemical format | Scientific Literature |
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