| # | Aladdin ID | Assay Type | Description | Organism | Compounds | Reference | BAO Format | Source | |
|---|---|---|---|---|---|---|---|---|---|
| 1. | ALA3423932 | F | Agonist activity at human wild-type KISS1R expressed in HEK293 cells assessed as induction of intracellular Ca2+ mobilization after 30 mins by Fluo4 NW Ca2+ assay | Homo sapiens | 17 | ALA3421632 | cell-based format | Scientific Literature | |
| 2. | ALA3423933 | A | Stability in Ile-de-France ewe serum assessed as intact compound level at 50 uM incubated for 6 hrs by HPLC method | Ovis aries | 6 | ALA3421632 | cell-free format | Scientific Literature | |
| 3. | ALA3423935 | F | Potency index, ratio of EC50 for KP10 to EC50 for compound for agonist activity at human wild-type KISS1R expressed in HEK293 cells assessed as induction of intracellular Ca2+ mobilization after 30 mins by Fluo4 NW Ca2+ assay | Homo sapiens | 1 | ALA3421632 | cell-based format | Scientific Literature | |
| 4. | ALA3423937 | F | Increase in total plasma LH level in anoestrus Ile-de-France ewe at 5 nmol, iv by radioimmunoassay | Ovis aries | 2 | ALA3421632 | organism-based format | Scientific Literature | |
| 5. | ALA3423938 | F | Increase in maximal amplitude of plasma LH level in anoestrus Ile-de-France ewe at 5 nmol, iv by radioimmunoassay (Rvb = 0.4 +/- 0.2 ng/ml) | Ovis aries | 1 | ALA3421632 | organism-based format | Scientific Literature | |
| 6. | ALA3423939 | F | Increase in duration of increase of plasma LH level in anoestrus Ile-de-France ewe at 5 nmol, iv by radioimmunoassay | Ovis aries | 2 | ALA3421632 | organism-based format | Scientific Literature | |
| 7. | ALA3423940 | F | Increase in maximal amplitude of plasma LH level in anoestrus Ile-de-France ewe at 1 to 15 nmol, iv by radioimmunoassay | Ovis aries | 2 | ALA3421632 | organism-based format | Scientific Literature | |
| 8. | ALA3423941 | F | Increase in time duration of increase of plasma LH level in anoestrus Ile-de-France ewe at 1 to 15 nmol, iv by radioimmunoassay | Ovis aries | 2 | ALA3421632 | organism-based format | Scientific Literature | |
| 9. | ALA3423942 | F | Increase in total plasma LH level in anoestrus Ile-de-France ewe at 1 to 15 nmol, iv by radioimmunoassay | Ovis aries | 2 | ALA3421632 | organism-based format | Scientific Literature | |
| 10. | ALA3423987 | F | Agonist activity at human NPFF1R expressed in CHO cells assessed as effect on forskolin-induced cAMP accumulation after 15 mins by luminescence based assay | Homo sapiens | 3 | ALA3421632 | cell-based format | Scientific Literature | |
| 11. | ALA3423988 | B | Selectivity index, ratio of EC50 for human NPFF1R to EC50 for human wild-type KISS1R | Homo sapiens | 3 | ALA3421632 | assay format | Scientific Literature |
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