| # | Aladdin ID | Assay Type | Description | Organism | Compounds | Reference | BAO Format | Source | |
|---|---|---|---|---|---|---|---|---|---|
| 1. | ALA3429766 | B | Inhibition of His-tagged human recombinant SIRT1 expressed in Escherichia coli using Cbz-Lys(Ac)-AMC as substrate by fluorescence assay | Homo sapiens | 13 | ALA3425433 | assay format | Scientific Literature | |
| 2. | ALA3429768 | B | Inhibition of His-tagged human recombinant SIRT2 expressed in Escherichia coli using Cbz-Lys(Ac)-AMC as substrate by fluorescence assay | Homo sapiens | 8 | ALA3425433 | assay format | Scientific Literature | |
| 3. | ALA3429770 | B | Inhibition of HDAC1 (unknown origin) | Homo sapiens | 36 | ALA3425433 | single protein format | Scientific Literature | |
| 4. | ALA3429771 | B | Inhibition of HDAC2 (unknown origin) | Homo sapiens | 36 | ALA3425433 | single protein format | Scientific Literature | |
| 5. | ALA3429772 | B | Inhibition of HDAC6 (unknown origin) | Homo sapiens | 36 | ALA3425433 | single protein format | Scientific Literature | |
| 6. | ALA3429773 | B | Inhibition of HDAC8 (unknown origin) | Homo sapiens | 36 | ALA3425433 | single protein format | Scientific Literature | |
| 7. | ALA3429777 | B | Inhibition of SIRT1-mediated endogenous p53 deacetylase activity in human Namalwa cells assessed as concentration required to enhance p53 deacetylation to twice the basal level after 3 hrs by ELISA | Homo sapiens | 7 | ALA3425433 | cell-based format | Scientific Literature | |
| 8. | ALA3429778 | A | Metabolic stability in mouse plasma | Mus musculus | 2 | ALA3425433 | cell-free format | Scientific Literature | |
| 9. | ALA3430204 | A | Clearance in rat | Rattus norvegicus | 2 | ALA3425433 | organism-based format | Scientific Literature | |
| 10. | ALA3430205 | A | Half life in rat | Rattus norvegicus | 2 | ALA3425433 | organism-based format | Scientific Literature | |
| 11. | ALA3430206 | A | Oral bioavailability in rat | Rattus norvegicus | 2 | ALA3425433 | organism-based format | Scientific Literature | |
| 12. | ALA3430207 | B | Inhibition of HDAC4 (unknown origin) | Homo sapiens | 35 | ALA3425433 | single protein format | Scientific Literature | |
| 13. | ALA3430208 | B | Inhibition of HDAC5 (unknown origin) | Homo sapiens | 35 | ALA3425433 | single protein format | Scientific Literature | |
| 14. | ALA3430209 | B | Inhibition of HDAC7 (unknown origin) | Homo sapiens | 35 | ALA3425433 | single protein format | Scientific Literature |
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