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| # | Aladdin ID | Assay Type | Description | Organism | Compounds | Reference | BAO Format | Source |
| 1. | ALA3541118 | F | Inhibition of MetAP2 level in Sprague-Dawley rat lymph nodes assessed as free enzyme level at 3 mg/kg, po by ELISA | Rattus norvegicus | 5 | | organism-based format | Scientific Literature |
| 2. | ALA3541119 | F | Inhibition of MetAP2 level in Sprague-Dawley rat thymus assessed as free enzyme level at 3 mg/kg, po by ELISA | Rattus norvegicus | 5 | | organism-based format | Scientific Literature |
| 3. | ALA3541120 | F | Inhibition of MetAP2 level in Sprague-Dawley rat whole blood assessed as free enzyme level at 3 mg/kg, po by ELISA | Rattus norvegicus | 5 | | organism-based format | Scientific Literature |
| 4. | ALA3539266 | F | Inhibition of MetAP2 level in Sprague-Dawley rat lung assessed as free enzyme level at 0.3 mg/kg, po by ELISA | Rattus norvegicus | 5 | | organism-based format | Scientific Literature |
| 5. | ALA3540061 | F | Inhibition of MetAP2 level in Sprague-Dawley rat liver assessed as free enzyme level at 0.3 mg/kg, po by ELISA | Rattus norvegicus | 5 | | organism-based format | Scientific Literature |
| 6. | ALA3540062 | F | Inhibition of MetAP2 level in Sprague-Dawley rat lymph nodes assessed as free enzyme level at 0.3 mg/kg, po by ELISA | Rattus norvegicus | 5 | | organism-based format | Scientific Literature |
| 7. | ALA3540063 | F | Inhibition of MetAP2 level in Sprague-Dawley rat thymus assessed as free enzyme level at 0.3 mg/kg, po by ELISA | Rattus norvegicus | 5 | | organism-based format | Scientific Literature |
| 8. | ALA3540064 | F | Inhibition of MetAP2 level in Sprague-Dawley rat whole blood assessed as free enzyme level at 0.3 mg/kg, po by ELISA | Rattus norvegicus | 5 | | organism-based format | Scientific Literature |
| 9. | ALA3540065 | F | Inhibition of MetAP2 level in Sprague-Dawley rat liver assessed as free enzyme level at 3 mg/kg, po by ELISA | Rattus norvegicus | 5 | | organism-based format | Scientific Literature |
| 10. | ALA3540066 | F | Inhibition of MetAP2 level in Sprague-Dawley rat liver assessed as free enzyme level at 0.3 mg/kg, iv by ELISA | Rattus norvegicus | 5 | | organism-based format | Scientific Literature |
| 11. | ALA3540067 | F | Inhibition of MetAP2 level in Sprague-Dawley rat lung assessed as free enzyme level at 3 mg/kg, po by ELISA | Rattus norvegicus | 5 | | organism-based format | Scientific Literature |
| 12. | ALA3527958 | B | Inhibition of human MetAP2 assessed as remaining enzyme activity after 8 hrs | Homo sapiens | 8 | | single protein format | Scientific Literature |
| 13. | ALA3527960 | B | Inhibition of human MetAP2 activity after end of experiment | Homo sapiens | 3 | | single protein format | Scientific Literature |
| 14. | ALA3527961 | B | Inhibition of MetAP2 activity in HUVEC assessed as inhibition of cell proliferation by MTT assay | Homo sapiens | 8 | | single protein format | Scientific Literature |
| 15. | ALA3527969 | A | Tmax in non-Hodgkin lymphoma patient treated with PPI-2458 at 15 mg, po alternate days for 21 days | Homo sapiens | 6 | | organism-based format | Scientific Literature |
| 16. | ALA3527970 | A | Cmax in non-Hodgkin lymphoma patient treated with PPI-2458 at 15 mg, po alternate days for 21 days | Homo sapiens | 6 | | organism-based format | Scientific Literature |
| 17. | ALA3527971 | A | AUC (0 to t hrs) in non-Hodgkin lymphoma patient treated with PPI-2458 at 15 mg, po alternate days for 21 days | Homo sapiens | 6 | | organism-based format | Scientific Literature |
| 18. | ALA3527972 | A | AUC (0 to infinity) in non-Hodgkin lymphoma patient treated with PPI-2458 at 15 mg, po alternate days for 21 days | Homo sapiens | 5 | | organism-based format | Scientific Literature |
| 19. | ALA3527973 | A | Half life in non-Hodgkin lymphoma patient treated with PPI-2458 at 15 mg, po alternate days for 21 days | Homo sapiens | 5 | | organism-based format | Scientific Literature |
| 20. | ALA3527974 | A | Retention time in human liver microsomes treated with at 5 mM PPI-2458 by LC/MS analysis | Homo sapiens | 4 | | assay format | Scientific Literature |