| # | Aladdin ID | Assay Type | Description | Organism | Compounds | Reference | BAO Format | Source | |
|---|---|---|---|---|---|---|---|---|---|
| 1. | ALA3588429 | B | Displacement of [3H]-PGE2 from rat EP2 receptor overexpressed in human ECV304 cell membranes by scintillation proximity assay | Rattus norvegicus | 2 | cell-based format | Scientific Literature | ||
| 2. | ALA3588430 | B | Displacement of [3H]-PGE2 from human EP2 receptor overexpressed in human ECV304 cell membranes by scintillation proximity assay | Homo sapiens | 54 | cell-based format | Scientific Literature | ||
| 3. | ALA3588431 | B | Displacement of [3H]-PGE2 from mouse EP2 receptor overexpressed in human ECV304 cell membranes by scintillation proximity assay | Mus musculus | 2 | cell-based format | Scientific Literature | ||
| 4. | ALA3588432 | B | Displacement of [3H]-PGE2 from human EP1 receptor overexpressed in human ECV304 cell membranes by scintillation proximity assay | Homo sapiens | 6 | cell-based format | Scientific Literature | ||
| 5. | ALA3588433 | B | Displacement of [3H]-PGE2 from human EP4 receptor overexpressed in human ECV304 cell membranes by scintillation proximity assay | Homo sapiens | 6 | cell-based format | Scientific Literature | ||
| 6. | ALA3588434 | B | Displacement of [3H]-PGE2 from human EP3 receptor overexpressed in human ECV304 cell membranes by scintillation proximity assay | Homo sapiens | 6 | cell-based format | Scientific Literature | ||
| 7. | ALA3588435 | F | Antagonist activity at human EP2 receptor overexpressed in human ECV304 cells assessed as inhibition of prostaglandin E2-induced cAMP production | Homo sapiens | 54 | cell-based format | Scientific Literature | ||
| 8. | ALA3588436 | F | Antagonist activity at rat EP2 receptor overexpressed in human ECV304 cells assessed as inhibition of prostaglandin E2-induced cAMP production | Rattus norvegicus | 2 | cell-based format | Scientific Literature | ||
| 9. | ALA3588437 | F | Antagonist activity at mouse EP2 receptor overexpressed in human ECV304 cells assessed as inhibition of prostaglandin E2-induced cAMP production | Mus musculus | 2 | cell-based format | Scientific Literature | ||
| 10. | ALA3588438 | A | Inhibition of CYP3A4 (unknown origin) at 3 uM relative to control | Homo sapiens | 19 | single protein format | Scientific Literature | ||
| 11. | ALA3588440 | A | Clearance in human liver microsomes at 10 uM by LC-MS analysis | Homo sapiens | 4 | assay format | Scientific Literature | ||
| 12. | ALA3588441 | A | Clearance in rat liver microsomes at 10 uM by LC-MS analysis | Rattus norvegicus | 4 | assay format | Scientific Literature | ||
| 13. | ALA3588444 | B | Selectivity ratio of IC50 for human EP4 receptor overexpressed in human ECV304 cell membranes to IC50 for human EP2 receptor overexpressed in human ECV304 cell membranes | Homo sapiens | 5 | cell-based format | Scientific Literature | ||
| 14. | ALA3588450 | F | Inhibition of human DP receptor assessed as LTD4-mediated intracellular calcium mobilization by cell-based aequorin luminescence assay | Homo sapiens | 1 | cell-based format | Scientific Literature | ||
| 15. | ALA3588451 | F | Inhibition of human IP receptor assessed as LTD4-mediated intracellular calcium mobilization by cell-based aequorin luminescence assay | Homo sapiens | 1 | cell-based format | Scientific Literature | ||
| 16. | ALA3588452 | F | Inhibition of human TP receptor assessed as LTD4-mediated intracellular calcium mobilization by call-based aequorin luminescence assay | Homo sapiens | 1 | cell-based format | Scientific Literature | ||
| 17. | ALA3588453 | F | Inhibition of human CRTH2 receptor assessed as LTD4-mediated intracellular calcium mobilization by cell-based aequorin luminescence assay | Homo sapiens | 1 | cell-based format | Scientific Literature | ||
| 18. | ALA3588454 | B | Selectivity ratio of IC50 for human DP receptor by cell-based aequorin luminescence assay to IC50 for human EP2 receptor overexpressed in human ECV304 cells by cAMP assay | Homo sapiens | 1 | cell-based format | Scientific Literature | ||
| 19. | ALA3588455 | B | Selectivity ratio of IC50 for human IP receptor by cell-based aequorin luminescence assay to IC50 for human EP2 receptor overexpressed in human ECV304 cells by cAMP assay | Homo sapiens | 1 | cell-based format | Scientific Literature | ||
| 20. | ALA3588456 | B | Selectivity ratio of IC50 for human TP receptor by cell-based aequorin luminescence assay to IC50 for human EP2 receptor overexpressed in human ECV304 cells by cAMP assay | Homo sapiens | 1 | cell-based format | Scientific Literature |
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