| # | Aladdin ID | Assay Type | Description | Organism | Compounds | Reference | BAO Format | Source | |
|---|---|---|---|---|---|---|---|---|---|
| 1. | ALA3587482 | B | Binding affinity to human OX2 receptor | Homo sapiens | 30 | ALA3585263 | single protein format | Scientific Literature | |
| 2. | ALA3587483 | B | Binding affinity to human OX1 receptor | Homo sapiens | 30 | ALA3585263 | single protein format | Scientific Literature | |
| 3. | ALA3587484 | B | Selectivity ratio of Ki for human OX1 receptor to Ki for human OX2 receptor | Homo sapiens | 1 | ALA3585263 | assay format | Scientific Literature | |
| 4. | ALA3587700 | A | Metabolic stability in rat liver microsomes assessed as extraction ratio at 1 uM measured over 1 hr by LC-MS/MS analysis | Rattus norvegicus | 12 | ALA3585263 | assay format | Scientific Literature | |
| 5. | ALA3587701 | A | Metabolic stability in human liver microsomes assessed as extraction ratio at 1 uM measured over 1 hr by LC-MS/MS analysis | Homo sapiens | 12 | ALA3585263 | assay format | Scientific Literature | |
| 6. | ALA3587702 | B | Inhibition of [3H]-astemizole binding to human ERG expressed in HEK293 cells | Homo sapiens | 12 | ALA3585263 | cell-based format | Scientific Literature | |
| 7. | ALA3587703 | B | Binding affinity to rat OX2 receptor | Rattus norvegicus | 12 | ALA3585263 | single protein format | Scientific Literature | |
| 8. | ALA3587704 | F | Ex vivo OX2 receptor occupancy in Sprague-Dawley rat brain at 10 mg/kg, po after 30 mins by autoradiographic analysis | Rattus norvegicus | 1 | ALA3585263 | organism-based format | Scientific Literature |
The page will load shortly, Thanks for your patience!