| # | Aladdin ID | Assay Type | Description | Organism | Compounds | Reference | BAO Format | Source | |
|---|---|---|---|---|---|---|---|---|---|
| 1. | ALA3588237 | Binding | Inhibition of BTK autophosphorylation in human Raji cells after 30 mins by Phos-Y223 Btk HTRF assay | Homo sapiens | 5 | ALA3585313 | cell-based format | Scientific Literature | |
| 2. | ALA3588238 | Binding | Inhibition of Lck (unknown origin) | Homo sapiens | 6 | ALA3585313 | single protein format | Scientific Literature | |
| 3. | ALA3588239 | ADME | Hepatic extraction ratio in human liver microsomes at 1 uM up to 30 mins by LC-MS/MS analysis | Homo sapiens | 5 | ALA3585313 | assay format | Scientific Literature | |
| 4. | ALA3588240 | ADME | Hepatic extraction ratio in rat liver microsomes at 1 uM up to 30 mins by LC-MS/MS analysis | Rattus norvegicus | 1 | ALA3585313 | assay format | Scientific Literature | |
| 5. | ALA3588241 | ADME | Apparent permeability across apical to basolateral side in pig LLC-PK1 cells expressing MDR1 | Sus scrofa | 1 | ALA3585313 | cell-based format | Scientific Literature | |
| 6. | ALA3588242 | ADME | Efflux ratio of apparent permeability across apical to basolateral side over basolateral to apical side in pig LLC-PK1 cells expressing MDR1 | Sus scrofa | 1 | ALA3585313 | cell-based format | Scientific Literature | |
| 7. | ALA3588243 | ADME | Clearance in Sprague-Dawley rat at 1 mg/kg, iv | Rattus norvegicus | 2 | ALA3585313 | organism-based format | Scientific Literature | |
| 8. | ALA3588244 | ADME | Hepatic extraction ratio in Sprague-Dawley rat at 1 mg/kg, iv | Rattus norvegicus | 1 | ALA3585313 | organism-based format | Scientific Literature | |
| 9. | ALA3588245 | ADME | Volume of distribution at steady state in Sprague-Dawley rat at 1 mg/kg, iv and 4 mg/kg, po | Rattus norvegicus | 2 | ALA3585313 | organism-based format | Scientific Literature | |
| 10. | ALA3588246 | ADME | Half life in Sprague-Dawley rat at 1 mg/kg, iv and 4 mg/kg, po | Rattus norvegicus | 2 | ALA3585313 | organism-based format | Scientific Literature | |
| 11. | ALA3588247 | ADME | Oral bioavailability in Sprague-Dawley rat at 4 mg/kg | Rattus norvegicus | 2 | ALA3585313 | organism-based format | Scientific Literature | |
| 12. | ALA3588253 | Binding | Inhibition of BTK in human Raji cells after 30 mins by HTRF assay | Homo sapiens | 6 | ALA3585313 | cell-based format | Scientific Literature | |
| 13. | ALA5252705 | Binding | Inhibition of NEK10 (unknown origin) at 1 uM relative to control | Homo sapiens | 43 | ALA5252509 | single protein format | Scientific Literature | |
| 14. | ALA5252734 | Binding | Inhibition of TIE2 (unknown origin) at 1 uM relative to control | Homo sapiens | 3 | ALA5252509 | single protein format | Scientific Literature | |
| 15. | ALA5252735 | Binding | Inhibition of BMX (unknown origin) at 1 uM relative to control | Homo sapiens | 3 | ALA5252509 | single protein format | Scientific Literature | |
| 16. | ALA5252736 | Binding | Inhibition of FGFR3 (unknown origin) at 1 uM relative to control | Homo sapiens | 3 | ALA5252509 | single protein format | Scientific Literature | |
| 17. | ALA5252737 | Binding | Inhibition of YSK4 (unknown origin) at 1 uM relative to control | Homo sapiens | 3 | ALA5252509 | single protein format | Scientific Literature | |
| 18. | ALA5252738 | Binding | Inhibition of BTK (unknown origin) at 1 uM relative to control | Homo sapiens | 3 | ALA5252509 | single protein format | Scientific Literature |
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