| # | Aladdin ID | Assay Type | Description | Organism | Compounds | Reference | BAO Format | Source | |
|---|---|---|---|---|---|---|---|---|---|
| 1. | ALA3591676 | B | Inhibition of JARID1A (unknown origin) using biotinylated H3K9mel peptide after 60 mins by Alpha screen assay | Homo sapiens | 17 | ALA3588787 | single protein format | Scientific Literature | |
| 2. | ALA3591677 | B | Inhibition of JMJD2C (unknown origin) using H3K9mel peptide | Homo sapiens | 17 | ALA3588787 | single protein format | Scientific Literature | |
| 3. | ALA3591678 | B | Inhibition of JMJD1A (unknown origin) using H3K9mel peptide | Homo sapiens | 17 | ALA3588787 | single protein format | Scientific Literature | |
| 4. | ALA3591679 | B | Inhibition of JHDM1F (unknown origin) using H3K9mel peptide | Homo sapiens | 17 | ALA3588787 | single protein format | Scientific Literature | |
| 5. | ALA3591681 | B | Inhibition of JARID1A overexpressed in human A549 cells assessed as H3K4me3/H3 ratio at 100 uM after 24 hrs by Western blot analysis | Homo sapiens | 4 | ALA3588787 | cell-based format | Scientific Literature | |
| 6. | ALA3591682 | B | Inhibition of JARID1A overexpressed in human A549 cells assessed as H3K4me3/H3 ratio at 300 uM after 24 hrs by Western blot analysis | Homo sapiens | 4 | ALA3588787 | cell-based format | Scientific Literature | |
| 7. | ALA3592268 | B | Inhibition of HDAC1 (unknown origin) at 100 uM | Homo sapiens | 3 | ALA3588787 | single protein format | Scientific Literature | |
| 8. | ALA4393226 | B | Inhibition of C-terminal FLAG-tagged human KDM5A expressed in Sf9 cells pre-incubated for 4 hrs before substrate addition and measured after 1 hr by AlphaScreen assay | Homo sapiens | 3 | ALA4392841 | cell-based format | Scientific Literature | |
| 9. | ALA4424780 | B | Inhibition of human C-terminal FLAG-tagged KDM5A (1 to 1090 residues) expressed in baculovirus infected Sf9 insect cells at 1 uM using H3(1-21)K4(Me3)-GGK(Biotin)/2-OG as substrate measured after 1 hr by Alphalisa assay relative to control | Homo sapiens | 6 | ALA4422684 | cell-based format | Scientific Literature | |
| 10. | ALA4424781 | B | Inhibition of human C-terminal FLAG-tagged KDM5A (1 to 1090 residues) expressed in baculovirus infected Sf9 insect cells at 25 uM using H3(1-21)K4(Me3)-GGK(Biotin)/2-OG as substrate measured after 1 hr by Alphalisa assay relative to control | Homo sapiens | 6 | ALA4422684 | cell-based format | Scientific Literature | |
| 11. | ALA4424782 | B | Inhibition of human C-terminal FLAG-tagged KDM5A (1 to 1090 residues) expressed in baculovirus infected Sf9 insect cells using H3(1-21)K4(Me3)-GGK(Biotin)/2-OG as substrate measured after 1 hr by Alphalisa assay | Homo sapiens | 7 | ALA4422684 | cell-based format | Scientific Literature | |
| 12. | ALA4424784 | B | Inhibition of human N-terminal FLAG/His-tagged KDM5B (2 to 751 residues) expressed in baculovirus infected Sf9 insect cells using H3(1-21)K4(Me3)-GGK(Biotin)/2-OG as substrate measured after 1 hr by Alphalisa assay | Homo sapiens | 4 | ALA4422684 | cell-based format | Scientific Literature | |
| 13. | ALA4424785 | B | Inhibition of full-length human N-terminal FLAG/His-tagged KDM5C (2 to 1560 residues) expressed in baculovirus infected Sf9 insect cells using H3(1-21)K4(Me3)-GGK(Biotin)/2-OG as substrate measured after 1 hr by Alphalisa assay | Homo sapiens | 4 | ALA4422684 | cell-based format | Scientific Literature | |
| 14. | ALA4424786 | B | Inhibition of human N-terminal FLAG/Avi-tagged KDM2A (2 to 700 residues) expressed in baculovirus infected Sf9 insect cells at 50 uM using H3(21-44)-K36(Me2)-GK(Biotin)/2-OG as substrate measured after 1 hr by Alphalisa assay relative to control | Homo sapiens | 4 | ALA4422684 | cell-based format | Scientific Literature | |
| 15. | ALA4424787 | B | Inhibition of human N-terminal FLAG/Avi-tagged KDM2A (2 to 700 residues) expressed in baculovirus infected Sf9 insect cells at 25 uM using H3(21-44)-K36(Me2)-GK(Biotin)/2-OG as substrate measured after 1 hr by Alphalisa assay relative to control | Homo sapiens | 4 | ALA4422684 | cell-based format | Scientific Literature | |
| 16. | ALA4424788 | B | Inhibition of human N-terminal FLAG-tagged KDM3A (2 to 1321 residues) expressed in baculovirus infected Sf9 insect cells at 50 uM using H3(1-21)K9(Me1)-GGK(Biotin)/2-OG as substrate measured after 1 hr by Alphalisa assay relative to control | Homo sapiens | 4 | ALA4422684 | cell-based format | Scientific Literature | |
| 17. | ALA4424789 | B | Inhibition of human N-terminal FLAG-tagged KDM3A (2 to 1321 residues) expressed in baculovirus infected Sf9 insect cells at 25 uM using H3(1-21)K9(Me1)-GGK(Biotin)/2-OG as substrate measured after 1 hr by Alphalisa assay relative to control | Homo sapiens | 4 | ALA4422684 | cell-based format | Scientific Literature | |
| 18. | ALA4424790 | B | Inhibition of human N-terminal His-tagged KDM4A (1 to 350 residues) expressed in Escherichia coli at 50 uM using H3(21-44)-K36(Me3)-GK(Biotin)/2-OG as substrate measured after 1 hr by Alphalisa assay relative to control | Homo sapiens | 4 | ALA4422684 | assay format | Scientific Literature | |
| 19. | ALA4424791 | B | Inhibition of human N-terminal His-tagged KDM4A (1 to 350 residues) expressed in Escherichia coli at 25 uM using H3(21-44)-K36(Me3)-GK(Biotin)/2-OG as substrate measured after 1 hr by Alphalisa assay relative to control | Homo sapiens | 4 | ALA4422684 | assay format | Scientific Literature | |
| 20. | ALA4424792 | B | Inhibition of human C-terminal FLAG-tagged KDM6B (1043 to end residues) expressed in baculovirus infected Sf9 insect cells at 50 uM using H3(21-44)-K27(Me3)-GK(Biotin)/2-OG as substrate measured after 1 hr by Alphalisa assay relative to control | Homo sapiens | 4 | ALA4422684 | cell-based format | Scientific Literature |
The page will load shortly, Thanks for your patience!