| # | Aladdin ID | Assay Type | Description | Organism | Compounds | Reference | BAO Format | Source | |
|---|---|---|---|---|---|---|---|---|---|
| 1. | ALA3592282 | B | Inhibition of SMYD2 (unknown origin) using biotinylated GSRAHSSHLKSKKGQSTSRH as substrate assessed as incorporation of tritium labeled methyl group from [3H]-SAM to biotinylated peptide substrate after 40 mins by scintillation proximity assay | Homo sapiens | 11 | single protein format | Scientific Literature | ||
| 2. | ALA3592283 | B | Competitive inhibition of SMYD2 (unknown origin) after 40 mins by scintillation proximity assay in presence of biotinylated GSRAHSSHLKSKKGQSTSRH substrate | Homo sapiens | 2 | single protein format | Scientific Literature | ||
| 3. | ALA3592284 | B | Uncompetitive inhibition of SMYD2 (unknown origin) after 40 mins by scintillation proximity assay in presence of SAM | Homo sapiens | 1 | single protein format | Scientific Literature | ||
| 4. | ALA3592285 | B | Inhibition of DNMT3A/3L (unknown origin) at 1 uM after 1 hr by filter-based assay | Homo sapiens | 1 | protein complex format | Scientific Literature | ||
| 5. | ALA3592286 | B | Inhibition of G9a (unknown origin) assessed as incorporation of tritium labeled methyl group from [3H]-SAM to substrate at 1 uM after 1 hr by scintillation proximity assay relative to control | Homo sapiens | 1 | single protein format | Scientific Literature | ||
| 6. | ALA3592287 | B | Inhibition of EHMT1 (unknown origin) assessed as incorporation of tritium labeled methyl group from [3H]-SAM to substrate at 1 uM after 1 hr by scintillation proximity assay relative to control | Homo sapiens | 1 | single protein format | Scientific Literature | ||
| 7. | ALA3592288 | B | Inhibition of SUV39H2 (unknown origin) assessed as incorporation of tritium labeled methyl group from [3H]-SAM to substrate at 1 uM after 1 hr by scintillation proximity assay relative to control | Homo sapiens | 1 | single protein format | Scientific Literature | ||
| 8. | ALA3592289 | B | Inhibition of SETDB1 (unknown origin) assessed as incorporation of tritium labeled methyl group from [3H]-SAM to substrate at 1 uM after 1 hr by scintillation proximity assay relative to control | Homo sapiens | 1 | single protein format | Scientific Literature | ||
| 9. | ALA3592290 | B | Inhibition of SETD7 (unknown origin) assessed as incorporation of tritium labeled methyl group from [3H]-SAM to substrate at 1 uM after 1 hr by scintillation proximity assay relative to control | Homo sapiens | 1 | single protein format | Scientific Literature | ||
| 10. | ALA3592291 | B | Inhibition of SETD8 (unknown origin) assessed as incorporation of tritium labeled methyl group from [3H]-SAM to substrate at 1 uM after 1 hr by scintillation proximity assay relative to control | Homo sapiens | 1 | single protein format | Scientific Literature | ||
| 11. | ALA3592398 | B | Inhibition of SUV420H1 (unknown origin) assessed as incorporation of tritium labeled methyl group from [3H]-SAM to substrate at 1 uM after 1 hr by scintillation proximity assay relative to control | Homo sapiens | 1 | single protein format | Scientific Literature | ||
| 12. | ALA3592399 | B | Inhibition of SUV420H2 (unknown origin) at 1 uM after 1 hr by filter-based assay | Homo sapiens | 1 | single protein format | Scientific Literature | ||
| 13. | ALA3592400 | B | Inhibition of MLL1 trimeric complex (unknown origin) assessed as incorporation of tritium labeled methyl group from [3H]-SAM to substrate at 1 uM after 1 hr by scintillation proximity assay relative to control | Homo sapiens | 1 | single protein format | Scientific Literature | ||
| 14. | ALA3592401 | B | Inhibition of EZH1 pentameric complex (unknown origin) assessed as incorporation of tritium labeled methyl group from [3H]-SAM to substrate at 1 uM after 1 hr by scintillation proximity assay relative to control | Homo sapiens | 1 | single protein format | Scientific Literature | ||
| 15. | ALA3592402 | B | Inhibition of EZH2 trimeric complex (unknown origin) assessed as incorporation of tritium labeled methyl group from [3H]-SAM to substrate at 1 uM after 1 hr by scintillation proximity assay relative to control | Homo sapiens | 1 | single protein format | Scientific Literature | ||
| 16. | ALA3592403 | B | Inhibition of SETD2 (unknown origin) assessed as incorporation of tritium labeled methyl group from [3H]-SAM to substrate at 1 uM after 1 hr by scintillation proximity assay relative to control | Homo sapiens | 1 | single protein format | Scientific Literature | ||
| 17. | ALA3592404 | B | Inhibition of PRDM9 (unknown origin) assessed as incorporation of tritium labeled methyl group from [3H]-SAM to substrate at 1 uM after 1 hr by scintillation proximity assay relative to control | Homo sapiens | 1 | single protein format | Scientific Literature | ||
| 18. | ALA3592405 | B | Inhibition of PRMT1 (unknown origin) assessed as incorporation of tritium labeled methyl group from [3H]-SAM to substrate at 1 uM after 1 hr by scintillation proximity assay relative to control | Homo sapiens | 1 | single protein format | Scientific Literature | ||
| 19. | ALA3592406 | B | Inhibition of PRMT3 (unknown origin) assessed as incorporation of tritium labeled methyl group from [3H]-SAM to substrate at 1 uM after 1 hr by scintillation proximity assay relative to control | Homo sapiens | 1 | single protein format | Scientific Literature | ||
| 20. | ALA3592407 | B | Inhibition of PRMT5-MEP50 complex (unknown origin) assessed as incorporation of tritium labeled methyl group from [3H]-SAM to substrate at 1 uM after 1 hr by scintillation proximity assay relative to control | Homo sapiens | 1 | protein complex format | Scientific Literature |
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