# | Aladdin ID | Assay Type | Description | Organism | Compounds | Reference | BAO Format | Source | |
---|---|---|---|---|---|---|---|---|---|
1. | ALA3599242 | B | Inhibition of human OGT using [3H]-UDP-GlcNAc as donor and recombinant nup2 as acceptor at 50 uM by liquid scintillation counting analysis | Homo sapiens | 8 | ALA3596110 | single protein format | Scientific Literature | |
2. | ALA3599243 | B | Inhibition of human OGT using [3H]-UDP-GlcNAc as donor and recombinant nup2 as acceptor by liquid scintillation counting analysis | Homo sapiens | 6 | ALA3596110 | single protein format | Scientific Literature | |
3. | ALA3599244 | B | Inhibition of human OGT using [3H]-UDP-GlcNAc as donor and recombinant nup2 as acceptor by Dixon plot analysis | Homo sapiens | 3 | ALA3596110 | single protein format | Scientific Literature | |
4. | ALA3599245 | B | Inhibition of OGT in human MCF7 cells assessed as decrease in intracellular O-GlcNAcylated protein level up to 500 uM after 24 to 48 hrs by immunoblot analysis | Homo sapiens | 7 | ALA3596110 | cell-based format | Scientific Literature | |
5. | ALA3599246 | B | Inhibition of OGT in human MCF10A cells assessed as decrease in intracellular O-GlcNAcylated protein level up to 500 uM after 24 to 48 hrs by immunoblot analysis | Homo sapiens | 1 | ALA3596110 | cell-based format | Scientific Literature | |
6. | ALA3599247 | B | Inhibition of OGT in human HeLa cells assessed as decrease in intracellular O-GlcNAcylated protein level up to 500 uM after 24 to 48 hrs by immunoblot analysis | Homo sapiens | 1 | ALA3596110 | cell-based format | Scientific Literature | |
7. | ALA3599248 | A | Permeability across POPC liposomes by out-in method | 2 | ALA3596110 | assay format | Scientific Literature | ||
8. | ALA3599249 | A | Permeability across POPC liposomes by in-out method | 2 | ALA3596110 | assay format | Scientific Literature |