| # | Aladdin ID | Assay Type | Description | Organism | Compounds | Reference | BAO Format | Source | |
|---|---|---|---|---|---|---|---|---|---|
| 1. | ALA3602662 | B | Displacement of [3H]-1-MeHis-TRH from mouse TRH-R1 expressed in HEK293 cells incubated up to 4 hrs by scintillation counting method | Mus musculus | 18 | ALA3600362 | cell-based format | Scientific Literature | |
| 2. | ALA3602663 | B | Displacement of [3H]-1-MeHis-TRH from mouse TRH-R2 expressed in HEK293 cells incubated up to 4 hrs by scintillation counting method | Mus musculus | 18 | ALA3600362 | cell-based format | Scientific Literature | |
| 3. | ALA3602664 | F | Agonist activity at mouse TRH-R1 expressed in HEK293 cells assessed as induction of changes in intracellular Ca2+ level by FLIPR method | Mus musculus | 18 | ALA3600362 | cell-based format | Scientific Literature | |
| 4. | ALA3602665 | F | Agonist activity at mouse TRH-R2 expressed in HEK293 cells assessed as induction of changes in intracellular Ca2+ level by FLIPR method | Mus musculus | 18 | ALA3600362 | cell-based format | Scientific Literature | |
| 5. | ALA3602666 | B | Selectivity index, ratio of EC50 for agonist activity at mouse TRH-R1 expressed in HEK293 cells to EC50 for agonist activity at mouse TRH-R2 expressed in HEK293 cells | Mus musculus | 18 | ALA3600362 | cell-based format | Scientific Literature | |
| 6. | ALA3602667 | F | Reduction in pentobarbital-induced sleeping time in Swiss mouse at 10 umol/kg, iv | Mus musculus | 18 | ALA3600362 | organism-based format | Scientific Literature |
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