| # | Aladdin ID | Assay Type | Description | Organism | Compounds | Reference | BAO Format | Source | |
|---|---|---|---|---|---|---|---|---|---|
| 1. | ALA625932 | A | Pharmacokinetic parameter :drug bound to plasma was reported | 9 | ALA1131523 | cell-free format | Scientific Literature | ||
| 2. | ALA630127 | P | Dissociation constant (KD) of the compound | 5 | ALA1128457 | small-molecule physicochemical format | Scientific Literature | ||
| 3. | ALA630098 | P | Partition coefficient (logP) | 28 | ALA1136781 | small-molecule physicochemical format | Scientific Literature | ||
| 4. | ALA629855 | A | Pharmacokinetic parameter :volume apparent of distribution was reported | 11 | ALA1131523 | organism-based format | Scientific Literature | ||
| 5. | ALA633319 | A | Pharmacokinetic parameter :half life in humans was reported | Homo sapiens | 11 | ALA1131523 | organism-based format | Scientific Literature | |
| 6. | ALA633442 | A | pA2 value is determined compared to standard H1-antagonists | 5 | ALA1128457 | assay format | Scientific Literature | ||
| 7. | ALA646122 | B | Compound is evaluated for in vitro receptor binding affinity against Alpha-1 adrenergic receptor | Cavia porcellus | 4 | ALA1128457 | protein format | Scientific Literature | |
| 8. | ALA664809 | A | Inhibition of human cytochrome P450 3A4 | 28 | ALA1136781 | single protein format | Scientific Literature | ||
| 9. | ALA685708 | F | Oral antiallergy activity in the guinea pig anaphylaxis (GPA) model, at a pretreatment time of 1 h | Cavia porcellus | 5 | ALA1124311 | organism-based format | Scientific Literature | |
| 10. | ALA685710 | F | Oral antiallergy activity in the guinea pig anaphylaxis (GPA) model, at a pretreatment time of 24 h; NT=Not tested | Cavia porcellus | 1 | ALA1124311 | organism-based format | Scientific Literature | |
| 11. | ALA685711 | F | Oral antiallergy activity in the guinea pig anaphylaxis (GPA) model of, at a pretreatment time of 6 h | Cavia porcellus | 1 | ALA1124311 | organism-based format | Scientific Literature | |
| 12. | ALA689046 | F | Compound was evaluated for inhibition of contraction in guinea pig ileum induced by leukotriene D4 (LTD4); Not active | Cavia porcellus | 1 | ALA1128421 | organism-based format | Scientific Literature | |
| 13. | ALA686175 | F | Compound was evaluated for antihistaminic activity against isolated guinea pig ileum. | Cavia porcellus | 12 | ALA1128421 | organism-based format | Scientific Literature | |
| 14. | ALA689686 | F | Inhibition of histamine-inducedcontraction of the isolated guinea-pig ileum | Cavia porcellus | 3 | ALA1125997 | organism-based format | Scientific Literature | |
| 15. | ALA691014 | F | K+ channel blocking activity in human embryonic kidney cells expressing HERG Kv11.1 | Homo sapiens | 17 | ALA1135758 | cell-based format | Scientific Literature | |
| 16. | ALA693825 | B | Compound is evaluated for in vitro receptor binding affinity against H1 receptor | Cavia porcellus | 4 | ALA1128457 | single protein format | Scientific Literature | |
| 17. | ALA693832 | B | Inhibitory activity against Tritiated [3H]- mepyramine binding to histamine H1 receptor in guinea pig cerebral cortex | Cavia porcellus | 5 | ALA1124311 | tissue-based format | Scientific Literature | |
| 18. | ALA698451 | B | Dissociation constant was determined against H1 receptor of guinea pig lung membranes using radioligand binding assays. | Cavia porcellus | 2 | ALA1128421 | tissue-based format | Scientific Literature | |
| 19. | ALA696934 | B | Inhibition of specific binding of [3H]mepyramine to Histamine 1 receptors in guinea-pig | Cavia porcellus | 3 | ALA1125997 | single protein format | Scientific Literature | |
| 20. | ALA691452 | F | Antagonism of the human histamine H1 receptor | 24 | ALA1150559 | assay format | Scientific Literature |
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