#	Aladdin ID	Assay Type	Description	Organism	Compounds	Reference	BAO Format	Source
1.	ALA3609987	B	Inhibition of EGFR L858R/T790M double mutant in human H1975 cells assessed as inhibition of phosphorylation at Y1068 after 2 hrs by sandwich ELISA method	Homo sapiens	6	ALA3608213	cell-based format	Scientific Literature
2.	ALA3609988	B	Inhibition of EGFR E746-A750 deletion mutant in human PC9 cells assessed as inhibition of phosphorylation at Y1068 after 2 hrs by sandwich ELISA method	Homo sapiens	6	ALA3608213	cell-based format	Scientific Literature
3.	ALA3609989	B	Inhibition of EGFR L858R mutant in human H3255 cells assessed as inhibition of phosphorylation at Y1068 after 2 hrs by sandwich ELISA method	Homo sapiens	6	ALA3608213	cell-based format	Scientific Literature
4.	ALA3609990	B	Inhibition of EGFR deletion/T790M mutant in human PC9-DRH cells assessed as inhibition of phosphorylation at Y1068 after 2 hrs by sandwich ELISA method	Homo sapiens	6	ALA3608213	cell-based format	Scientific Literature
5.	ALA3609991	B	Inhibition of wild type EGFR in human A549 cells assessed as inhibition of phosphorylation at Y1068 after 2 hrs by sandwich ELISA method	Homo sapiens	6	ALA3608213	cell-based format	Scientific Literature
6.	ALA4178350	A	Inhibition of EGF-stimulated wild-type EGFR phosphorylation in human A549 cells preincubated for 2 hrs followed by EGF stimulation for 10 mins by sandwich ELISA	Homo sapiens	21	ALA4177539	cell-based format	Scientific Literature
7.	ALA4178351	B	Inhibition of EGFR T790M/L858R double mutant phosphorylation in human H1975 cells preincubated for 2 hrs followed by EGF stimulation for 10 mins by sandwich ELISA	Homo sapiens	22	ALA4177539	cell-based format	Scientific Literature
8.	ALA4178352	B	Selectivity index, ratio of IC50 for wild-type EGFR autophosphorylation in human A549 cells to IC50 for EGFR T790M/L858R double mutant autophosphorylation in human H1975 cells	Homo sapiens	15	ALA4177539	cell-based format	Scientific Literature
9.	ALA4178353	P	Lipophilicity, log D of the compound		16	ALA4177539	small-molecule physicochemical format	Scientific Literature
10.	ALA4178355	P	Glutathione reactivity of the compound in pH 7.4 phosphate buffer assessed as half life at 1 uM up to 120 mins by LC-MS/MS analysis relative to canertinib		15	ALA4177539	small-molecule physicochemical format	Scientific Literature
11.	ALA4178356	B	Inhibition of EGFR T790M/L858R double mutant (unknown origin)	Homo sapiens	23	ALA4177539	single protein format	Scientific Literature
12.	ALA4178358	A	Intrinsic clearance in human liver microsomes at 1 uM up to 45 mins in presence of NADPH by LC-MS/MS analysis	Homo sapiens	8	ALA4177539	microsome format	Scientific Literature
13.	ALA4178360	B	Inhibition of EGFR T790M/exon 19 deletion mutant phosphorylation in human PC9-DRH cells preincubated for 2 hrs followed by EGF stimulation for 10 mins by sandwich ELISA	Homo sapiens	10	ALA4177539	cell-based format	Scientific Literature
14.	ALA4178361	B	Inhibition of EGFR exon 19 deletion mutant phosphorylation in human PC9 cells preincubated for 2 hrs followed by EGF stimulation for 10 mins by sandwich ELISA	Homo sapiens	10	ALA4177539	cell-based format	Scientific Literature
15.	ALA4178362	B	Inhibition of EGFR L858R mutant phosphorylation in human H3255 cells preincubated for 2 hrs followed by EGF stimulation for 10 mins by sandwich ELISA	Homo sapiens	10	ALA4177539	cell-based format	Scientific Literature
16.	ALA4178363	B	Selectivity index, ratio of IC50 for wild-type EGFR autophosphorylation in human A549 cells to IC50 for EGFR exon 19 deletion mutant autophosphorylation in human PC9 cells	Homo sapiens	5	ALA4177539	cell-based format	Scientific Literature
17.	ALA4178437	B	Inhibition of EGFR T790M/L858R double mutant (unknown origin) assessed as ratio of observed rate constant to inhibitor concentration at 0.05 uM	Homo sapiens	1	ALA4177539	single protein format	Scientific Literature