| # | Aladdin ID | Assay Type | Description | Organism | Compounds | Reference | BAO Format | Source | |
|---|---|---|---|---|---|---|---|---|---|
| 1. | ALA3615682 | B | Inhibition of ROMK (unknown origin) expressed in HEK293 cells by thallium flux assay | Homo sapiens | 32 | ALA3612018 | cell-based format | Scientific Literature | |
| 2. | ALA3615683 | B | Displacement of [35S]-MK499 from human ERG expressed in HEK293 cells | Homo sapiens | 30 | ALA3612018 | cell-based format | Scientific Literature | |
| 3. | ALA3615685 | B | Selectivity ratio of IC50 for human ERG to IC50 for ROMK (unknown origin) | Homo sapiens | 17 | ALA3612018 | assay format | Scientific Literature | |
| 4. | ALA3615686 | B | Inhibition of human ERG expressed in HEK293 cells by electrophysiology assay | Homo sapiens | 8 | ALA3612018 | cell-based format | Scientific Literature | |
| 5. | ALA3615691 | A | Dose normalized AUC in Sprague-Dawley rat at 2 mg/kg, po | Rattus norvegicus | 9 | ALA3612018 | organism-based format | Scientific Literature | |
| 6. | ALA3615693 | A | Oral bioavailability in Sprague-Dawley rat at 2 mg/kg | Rattus norvegicus | 9 | ALA3612018 | organism-based format | Scientific Literature | |
| 7. | ALA3615694 | B | Inhibition of ROMK (unknown origin) expressed in HEK293 cells by electrophysiology assay | Homo sapiens | 7 | ALA3612018 | cell-based format | Scientific Literature | |
| 8. | ALA3615695 | B | Selectivity ratio of IC50 for human ERG by electrophysiology assay to IC50 for ROMK (unknown origin) by electrophysiology assay | Homo sapiens | 7 | ALA3612018 | assay format | Scientific Literature | |
| 9. | ALA3615696 | T | Cardiotoxicity in guinea pig assessed as change in QT interval at 2 mg/kg, iv | Cavia porcellus | 1 | ALA3612018 | organism-based format | Scientific Literature | |
| 10. | ALA3615697 | A | Unbound plasma concentration in guinea pig at 2 mg/kg, iv | Cavia porcellus | 1 | ALA3612018 | organism-based format | Scientific Literature | |
| 11. | ALA3615698 | A | Clearance in Sprague-Dawley rat at 1 mg/kg, iv and 2 mg/kg, po | Rattus norvegicus | 5 | ALA3612018 | organism-based format | Scientific Literature | |
| 12. | ALA3615699 | A | Half life in Sprague-Dawley rat at 1 mg/kg, iv and 2 mg/kg, po | Rattus norvegicus | 5 | ALA3612018 | organism-based format | Scientific Literature | |
| 13. | ALA3615700 | B | Inhibition of Kir2.3 potassium channel (unknown origin) | Homo sapiens | 1 | ALA3612018 | single protein format | Scientific Literature | |
| 14. | ALA3615701 | B | Inhibition of Kir2.1 potassium channel (unknown origin) | Homo sapiens | 1 | ALA3612018 | single protein format | Scientific Literature | |
| 15. | ALA3615702 | B | Inhibition of Kir4.1 potassium channel (unknown origin) | Homo sapiens | 1 | ALA3612018 | single protein format | Scientific Literature | |
| 16. | ALA3615703 | B | Inhibition of Kir7.1 potassium channel (unknown origin) | Homo sapiens | 1 | ALA3612018 | single protein format | Scientific Literature | |
| 17. | ALA3615704 | B | Inhibition of Nav1.2 channel (unknown origin) | Homo sapiens | 1 | ALA3612018 | single protein format | Scientific Literature | |
| 18. | ALA3615705 | B | Inhibition of Nav2.1 channel (unknown origin) | Homo sapiens | 1 | ALA3612018 | single protein format | Scientific Literature | |
| 19. | ALA3615706 | A | Inhibition of CYP3A4 (unknown origin) | Homo sapiens | 1 | ALA3612018 | single protein format | Scientific Literature | |
| 20. | ALA3615707 | A | Inhibition of CYP2D6 (unknown origin) | Homo sapiens | 1 | ALA3612018 | single protein format | Scientific Literature |
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